Compile Data Set for Download or QSAR
Found 90 of ec50 for UniProtKB: P43354
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50196291(6-(benzo[d][1,3]dioxol-5-yl)-5-methyl-3-phenylisox...)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371201(CHEMBL399807)copy SMILEScopy InChI
Affinity DataEC50:  3.5nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371206(CHEMBL401032)copy SMILEScopy InChI
Affinity DataEC50:  3.90nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50196289(6-(4-methoxyphenyl)-5-methyl-3-phenylisoxazolo[4,5...)copy SMILEScopy InChI
Affinity DataEC50:  4.10nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517820(CHEMBL4473232)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50580049(CHEMBL5086921)copy SMILES
Affinity DataEC50:  24nMAssay Description:Agonist activity at full length NURR1 (unknown origin) expressed in mouse MND9 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0K0DPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517810(CHEMBL4579076)copy SMILEScopy InChI
Affinity DataEC50:  25nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371210(CHEMBL247879)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371205(CHEMBL393713)copy SMILEScopy InChI
Affinity DataEC50:  31.9nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517819(CHEMBL4475176)copy SMILEScopy InChI
Affinity DataEC50:  38nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517811(CHEMBL4576867)copy SMILEScopy InChI
Affinity DataEC50:  45nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371209(CHEMBL246654)copy SMILEScopy InChI
Affinity DataEC50:  59.2nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517814(CHEMBL4461137)copy SMILEScopy InChI
Affinity DataEC50:  75nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371208(ISOXAZOLOPYRIDINONE)copy SMILEScopy InChI
Affinity DataEC50:  77.5nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517837(CHEMBL4455501)copy SMILEScopy InChI
Affinity DataEC50:  87nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371204(CHEMBL247478)copy SMILEScopy InChI
Affinity DataEC50:  113nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM86707(CAS_147511-69-1 | Pitavastatin)copy SMILEScopy InChI
Affinity DataEC50:  120nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6PD2PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371202(CHEMBL393714)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517833(CHEMBL4472621)copy SMILEScopy InChI
Affinity DataEC50:  140nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517832(CHEMBL4564985)copy SMILEScopy InChI
Affinity DataEC50:  218nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517814(CHEMBL4461137)copy SMILEScopy InChI
Affinity DataEC50:  219nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517814(CHEMBL4461137)copy SMILEScopy InChI
Affinity DataEC50:  219nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517817(CHEMBL4446736)copy SMILEScopy InChI
Affinity DataEC50:  323nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517809(CHEMBL4587411)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517812(CHEMBL4454933)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517813(CHEMBL4464547)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517815(CHEMBL4559712)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517816(CHEMBL4440984)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517818(CHEMBL4453694)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517821(CHEMBL4521080)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517822(CHEMBL4450849)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517823(CHEMBL4435806)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517824(CHEMBL4455780)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517825(CHEMBL4473547)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517826(CHEMBL4453191)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517827(CHEMBL4528015)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517830(CHEMBL4475835)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517844(CHEMBL4521819)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517846(CHEMBL4441108)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517847(CHEMBL4451443)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517828(CHEMBL4465777)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517829(CHEMBL4542579)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517831(CHEMBL4516628)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517851(CHEMBL4440924)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517843(CHEMBL4546699)copy SMILEScopy InChI
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50571364(CHEMBL4856824)copy SMILES
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at Gal4-fused human Nurr1 LBD expressed in HEK293T cells co-expressing firefly luciferase assessed as luciferase activity incubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60SV3PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM86704(CAS_93957-54-1 | Fluvastatin | cid_446155)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6PD2PubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371203(CHEMBL247263)copy SMILEScopy InChI
Affinity DataEC50: >2.00E+3nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50371207(CHEMBL247676)copy SMILEScopy InChI
Affinity DataEC50: >2.00E+3nMAssay Description:Activation of Nurr1 expressed in MN9D cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9J2RPubMed
TargetNuclear receptor subfamily 4 group A member 2(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50517836(CHEMBL4542143)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at full-length Gal4-fused NOT (unknown origin) expressed in CHO cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2SB9PubMed
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