Compile Data Set for Download or QSAR
Found 3 of ec50 for UniProtKB: P37172
TargetActivin receptor type-1(Mus musculus)
National Center for Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50466183(CHEMBL4283638)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Inhibition of BMP6-induced ALK2 transcriptional activity in mouse C2C12 cells expressing BRE-Luc after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8BBTPubMed
TargetActivin receptor type-1(Mus musculus)
National Center for Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50262079(4-(6-(4-(piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyri...)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Inhibition of BMP6-induced ALK2 transcriptional activity in mouse C2C12 cells expressing BRE-Luc after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetActivin receptor type-1(Mus musculus)
National Center for Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50466190(CHEMBL4288921)copy SMILEScopy InChI
Affinity DataEC50:  91nMAssay Description:Inhibition of BMP6-induced ALK2 transcriptional activity in mouse C2C12 cells expressing BRE-Luc after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8BBTPubMed