Compile Data Set for Download or QSAR
Found 2 of ic50 for UniProtKB: P42336
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/beta isoform(Homo sapiens (Human))
University of California, San Francisco

LigandPNGBDBM36408(1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1H-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP22S9PubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/beta isoform(Homo sapiens (Human))
University of California, San Francisco

LigandPNGBDBM36408(1-cyclobutyl-3-(3,4-dimethoxyphenyl)-1H-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of PI3K enzyme activity is measured in a microtiter plate-based fluorescence polarization (FP) assay.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP22S9PubMed