Compile Data Set for Download or QSAR
Found 6 of ic50 for UniProtKB: P43143
LigandPNGBDBM50516340(CHEMBL4439678)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77P3PubMed
LigandPNGBDBM50567426(CHEMBL4878856)copy SMILES
Affinity DataIC50: 23nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77P3PubMed
LigandPNGBDBM50567413(CHEMBL4865365)copy SMILES
Affinity DataIC50: 27nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77P3PubMed
LigandPNGBDBM50516342(CHEMBL4461998)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77P3PubMed
LigandPNGBDBM50445326(CHEMBL3104239)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Antagonist activity at rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of Ach-induced response at -70 mV holding pot...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ7231PubMed
LigandPNGBDBM50445326(CHEMBL3104239)copy SMILEScopy InChI
Affinity DataIC50: 222nMAssay Description:Inhibition of rat alpha6beta4 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current response measured aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN77P3PubMed