Compile Data Set for Download or QSAR
Found 9 of ic50 for UniProtKB: P29275
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182282(CHEMBL3818905)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41GQPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182281(CHEMBL3818205)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41GQPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182283(CHEMBL3819313)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41GQPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182284(CHEMBL3818888)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41GQPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41GQPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM21173(1,3-dipropyl-8-cyclopentylxanthine | 8-cyclopentyl...)copy SMILEScopy InChI
Affinity DataIC50: 656nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4W31
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50287703((E)-1-[(S)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4W31
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50368346(CHEMBL608008)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+4nMAssay Description:Maximal NECA stimulation of adenylate cyclase via Adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2M9098MPubMed
TargetAdenosine receptor A2a/A2b(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50079652((E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4W31