Compile Data Set for Download or QSAR
Found 41 of ic50 for UniProtKB: P09216
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108296(CHEMBL289772 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280871(12-(3-azidopropyl)-13-methyl-6,7,12,13-tetrahydro-...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280875(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128287(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-methyl-piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128282(3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128280(3-[1-(1-Ethyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108291(CHEMBL36891 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 222nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128286(3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128290(3-[1-(1-Cyclopropylmethyl-piperidin-4-yl)-1H-indol...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128281(18-dimethylaminomethyl-(18S)-17-oxa-4,14,21-triaza...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108299(CHEMBL288229 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128288(3-(1-Methyl-1H-indol-3-yl)-4-(1-piperidin-4-yl-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108295(CHEMBL288817 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280878(12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50052039(18-hydroxymethyl-(18S)-17-oxa-4,14,21-triazahexacy...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50MXM
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280874(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 590nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM2581(3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^{4,9}.0^...)copy SMILEScopy InChI
Affinity DataIC50: 680nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128285(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108297(CHEMBL288816 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108300(CHEMBL38338 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108293(CHEMBL277817 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128283(3-[1-(1-Benzyl-pyrrolidin-3-yl)-1H-indol-3-yl]-4-(...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50212623(CHEMBL299248)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50128284(3-(1-(1-benzylpiperidin-4-yl)-1H-indol-3-yl)-4-(1-...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319V87PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50285193(17-hydroxymethyl-18-oxa-4,14,22-triazahexacyclo[20...)copy SMILEScopy InChI
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50MXM
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108298(CHEMBL29709 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50212624(CHEMBL294684)copy SMILEScopy InChI
Affinity DataIC50: 8.10E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108292(CHEMBL37529 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50108294(CHEMBL288818 | Indolocarbazole analogue)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity for Growth factor receptor bound protein 2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2571B94PubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa-Hakko Kogyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50280867(2-(6,13-dimethyl-5-oxo-6,7,12,13-tetrahydro-5H-ind...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC03DJ