Compile Data Set for Download or QSAR
Found 15 of ic50 for UniProtKB: P31646
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of high affinity neuronal GABA uptake by synaptosomes of rat brain membraneMore data for this Ligand-Target Pair
LigandPNGBDBM24183(4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
LigandPNGBDBM50021186(4-Amino-3-hydroxy-butyric acid | CHEMBL296263 | S(...)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+4nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed
LigandPNGBDBM50021187(4-Amino-3-hydroxy-butyric acid | CHEMBL290216 | R(...)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed
LigandPNGBDBM50021189(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL40...)copy SMILEScopy InChI
Affinity DataIC50: 7.00E+4nMAssay Description:In vivo inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed
LigandPNGBDBM50225363(CHEMBL40363)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed
LigandPNGBDBM50021262(4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-5-ium-3-...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM50224812(CHEBI:35010 | CHEMBL170539)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM50224810(CHEMBL171241)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed
LigandPNGBDBM50224811(CHEMBL170753)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM50224809(CHEBI:34373 | Gaboxadol | LU-02030 | MK-0928)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM50224808(CHEMBL309689)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:In vitro effect on GABA uptake in a crude preparation of synaptosomes from rat brain.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P84CGXPubMed
LigandPNGBDBM50021185(5-Aminomethyl-4,5-dihydro-isoxazol-3-ol | CHEMBL42...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:In vitro inhibition of GABA uptake in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94NZPubMed