Compile Data Set for Download or QSAR
Found 255 of ic50 for UniProtKB: P03372
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521421(6-(2,4- dichlorophenyl)- 1-fluoro-5-[6- [(3S)-1-(3...)copy SMILES
Affinity DataIC50: 4nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521334(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 4nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521345(4-(2-fluoro-4- hydroxy- phenyl)-5-[4- [(3S)-1-(3- ...)copy SMILES
Affinity DataIC50: 5nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521255(3-(6-ethoxy-2- fluoro-3- pyridyl)-4-[6- [(3S)-1-(3...)copy SMILES
Affinity DataIC50: 6nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521360(4-(benzofuran- 5-yl)-5-[4-[(3S)- 1-(3- fluoropropy...)copy SMILES
Affinity DataIC50: 6nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521416(6-(6-ethoxy-2- fluoro-3- pyridyl)-5-[6- [(3S)-1-(3...)copy SMILES
Affinity DataIC50: 6nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521262(6-(6-ethoxy-2- fluoro-3- pyridyl)-5-[4- [[(3S)-1-(...)copy SMILES
Affinity DataIC50: 7nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521413(6-(2-fluoro-4- methyl-phenyl)- 5-[6-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 7nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521296(4-(benzofuran- 5-yl)-5-[4-[(3S)- 1-(3- fluoropropy...)copy SMILES
Affinity DataIC50: 7nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521384(4-(6-ethoxy-2- fluoro-3- pyridyl)-5-[6- [(3S)-1-(3...)copy SMILES
Affinity DataIC50: 7nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521374(4-(2,2- dimethylindolin- 5-yl)-5-[4-[(3S)- 1-(3- f...)copy SMILES
Affinity DataIC50: 8nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521428(6-(6-ethoxy-2- fluoro-3- pyridyl)-1- fluoro-5-[6- ...)copy SMILES
Affinity DataIC50: 8nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521418(6-(2,2- dimethylindolin- 5-yl)-5-[6-[(3S)- 1-(3- f...)copy SMILES
Affinity DataIC50: 9nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521383(4-[4- (difluoromethoxy)- 3-fluoro- phenyl]-5-[6- [...)copy SMILES
Affinity DataIC50: 9nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521354(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521295(4-(4-ethoxy-2- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521270(4-(2-fluoro-4- hydroxy- phenyl)-5-[4- [(3S)-1-(3- ...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521267(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521341(4-(4-fluoro-2- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 11nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521336(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521182(7-(2-fluoro-4- hydroxy- phenyl)-8-[4- [(3S)-1-(3- ...)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521415(6-(2,4- dichlorophenyl)- 5-[6-[(3S)-1-(3- fluoropr...)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521340(4-(2-fluoro-4- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521382(4-(2-chloro-4- methyl-phenyl)- 5-[6-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 13nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521344(4-(2-chloro-3- fluoro-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 14nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521378(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 15nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521192(3-(2-fluoro-4- methyl-phenyl)- 4-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 16nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521381(4-(2,4- dichlorophenyl)- 5-[(6-[(3S)-1-(3- fluorop...)copy SMILES
Affinity DataIC50: 16nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521335(4-(2-chloro-4- fluoro-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 17nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521373(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 20nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521362(4-(4-ethoxy-2- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 21nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521377(4-(2,2-dimethyl- 3H-benzofuran- 5-yl)-5-[4-[(3S)- ...)copy SMILES
Affinity DataIC50: 21nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521261(6-(2,4- dichlorophenyl)- 5-[4-[[(3S)-1- (3- fluoro...)copy SMILES
Affinity DataIC50: 21nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521195(4-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 23nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521380(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521425(6-[4- (difluoromethoxy)- 3-fluoro- phenyl]-1- fluo...)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521348(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521339(4-(3-chloro-2- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521338(4-(4-chloro-3- methyl-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 24nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521394(4-[4- (fluoromethoxy) phenyl]-5-[4- [(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 25nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521369(4-(2,2-difluoro- 1,3- benzodioxol-5- yl)-5-[4-[(3S...)copy SMILES
Affinity DataIC50: 25nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521343(4-(4-chloro-2- fluoro-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 26nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521417(6-[4- (difluoromethoxy)- 3-fluoro- phenyl]-5-[6- [...)copy SMILES
Affinity DataIC50: 27nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521297(4-(2-fluoro-4- methoxy- phenyl)-5-[4- [(3S)-1-(3- ...)copy SMILES
Affinity DataIC50: 27nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521198(3-(2-chloro-4- fluoro-phenyl)- 4-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 27nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521352(5-[4-[(3S)-1-(3- fluoropropyl)pyr- rolidin-3- yl]o...)copy SMILES
Affinity DataIC50: 28nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521254(3-(2-fluoro-4- methyl-phenyl)- 4-[6-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 29nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521297(4-(2-fluoro-4- methoxy- phenyl)-5-[4- [(3S)-1-(3- ...)copy SMILES
Affinity DataIC50: 31nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521337(4-(4-chloro-3- fluoro-phenyl)- 5-[4-[(3S)-1-(3- fl...)copy SMILES
Affinity DataIC50: 31nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
TargetEstrogen receptor [298-554,D538G](Homo sapiens (Human))TBA
LigandPNGBDBM521282(9-fluoro-4-(2- fluoro-4-methyl- phenyl)-5-[4- [(3S...)copy SMILES
Affinity DataIC50: 31nMAssay Description:Antagonistic potency of compounds was evaluated using LanthaScreenŽ TR-FRET ERα Coactivator Assay (ThermoFisher) with modifications. It is a com...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ8BT3US Patent
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