Compile Data Set for Download or QSAR
Found 16 of ic50 for UniProtKB: P29702
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13361((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 100nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13373((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 600nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMedMMDB
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13358((2S)-2-{[(2R)-1-[(2S)-2-[(2R)-2-amino-3-sulfanylpr...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13359((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13363((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13362((2S)-2-[(2R)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13360((2S)-2-[(2R)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13365((2S)-2-[(2S)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13369((2S)-2-[(2S)-3-(4-hydroxy-2,5-dimethylphenyl)-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 5.50E+3nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13370((2S)-2-[(2R)-3-(4-hydroxy-2,5-dimethylphenyl)-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13367((2S)-2-[(2S)-3-(4-hydroxy-2,3-dimethylphenyl)-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13364((2S)-2-[(2R)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13366((2S)-2-[(2R)-2-[(2S)-2-[(2R)-2-amino-3-sulfanylpro...)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13371(CAAX Analogue 14 | Compound XIV | methyl (2S)-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 2.04E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13372(CAAX Analogue 15 | Compound XV | methyl (2S)-2-[(2...)copy SMILEScopy InChI
Affinity DataIC50: 7.05E+4nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Universita di Napoli Federico II

LigandPNGBDBM13368((2S)-2-[(2R)-3-(4-hydroxy-2,3-dimethylphenyl)-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 7.5 T: 2°CAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22V2DCHPubMed