Compile Data Set for Download or QSAR
Found 23 of ic50 for UniProtKB: P32240
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606234(CHEMBL5189703)copy SMILES
Affinity DataIC50: 2.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520104(CHEMBL4535971)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606218(CHEMBL5181722)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606245(CHEMBL5186525)copy SMILES
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520097(CHEMBL4564092)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606219(CHEMBL5179032)copy SMILES
Affinity DataIC50: 29nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520100(CHEMBL4576681)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520098(CHEMBL4548291)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606223(CHEMBL5195058)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520071(CHEMBL4440382)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606226(CHEMBL5188328)copy SMILES
Affinity DataIC50: 67nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520073(CHEMBL4591792)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50537002(CHEMBL4483026)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Antagonist activity at mouse EP4R assessed as inhibition of agonist-induced cAMP production by fluorescent cAMP tracer cAMP-d2 based FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7KSBPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM119448(US8686018, 107)copy SMILEScopy InChI
Affinity DataIC50: 101nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50537004(CHEMBL4584103)copy SMILEScopy InChI
Affinity DataIC50: 113nMAssay Description:Antagonist activity at mouse EP4R assessed as inhibition of agonist-induced cAMP production by fluorescent cAMP tracer cAMP-d2 based FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7KSBPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520103(CHEMBL4455965)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520101(CHEMBL4439228)copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520069(CHEMBL4457944)copy SMILEScopy InChI
Affinity DataIC50: 135nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM119448(US8686018, 107)copy SMILEScopy InChI
Affinity DataIC50: 181nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520072(CHEMBL4550862)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50606233(CHEMBL5208220)copy SMILES
Affinity DataIC50: 336nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM8CD4PubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520102(CHEMBL4453648)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed
TargetProstaglandin E2 receptor EP4 subtype(Mus musculus (Mouse))TBA
LigandPNGBDBM50520086(CHEMBL4463343)copy SMILEScopy InChI
Affinity DataIC50: 906nMAssay Description:Antagonist activity at mouse EP4 expressed in CHO cells coexpressing G16-alpha assessed as intracellular calcium flux preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58QRTPubMed