Compile Data Set for Download or QSAR
Found 12 of ic50 for UniProtKB: P52732
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36351(CID148124 | Docetaxel)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36351(CID148124 | Docetaxel)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36351(CID148124 | Docetaxel)copy SMILEScopy InChI
Affinity DataIC50: 0.350nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36350(6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-qu...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36351(CID148124 | Docetaxel)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36350(6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-qu...)copy SMILEScopy InChI
Affinity DataIC50: 0.830nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36350(6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-qu...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM36350(6-[4-(Trifluoromethyl)phenyl]-3,4-dihydro-2(1H)-qu...)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM50220156((R)-N-(3-aminopropyl)-N-(1-(3-benzyl-7-chloro-4-ox...)copy SMILEScopy InChI
Affinity DataIC50: 87.3nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM50220156((R)-N-(3-aminopropyl)-N-(1-(3-benzyl-7-chloro-4-ox...)copy SMILEScopy InChI
Affinity DataIC50: 675nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM50220156((R)-N-(3-aminopropyl)-N-(1-(3-benzyl-7-chloro-4-ox...)copy SMILEScopy InChI
Affinity DataIC50: 903nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed
TargetKinesin-like protein KIF11 [D130V](Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM50220156((R)-N-(3-aminopropyl)-N-(1-(3-benzyl-7-chloro-4-ox...)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+3nMpH: 6.8Assay Description:Cell proliferation assay for ispinesib-resistant DCT116-D130V cellMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0DHCPubMed