Compile Data Set for Download or QSAR
Found 8 of ic50 for UniProtKB: P19492
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50316374(CHEMBL1096289 | N-(4-hydroxyphenylpropanyl)-spermi...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of rat recombinant GluA3 receptor expressed in Xenopus oocytes assessed as inhibition of 300 uM kainate-induced currentMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6CB2PubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50355329(CHEMBL1835336)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at recombinant rat GluA3 flip isoform receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced cu...More data for this Ligand-Target Pair
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50158561(2-[3-(3-bromophenyl)ureido]-4-chlorobenzenesulfoni...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50158556(1-(3-bromophenyl)-3-[5-chloro-2-(1H-tetrazol-5-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50158555(1-[5-chloro-2-(5-oxo-4,5-dihydro-[1,2,4]oxadiazol-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50137125(2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50137124(4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed
TargetGlutamate receptor 3(RAT)
University of California

Curated by ChEMBL
LigandPNGBDBM50158554(CHEMBL224688 | {2-[3-(3-bromophenyl)ureido]-4-chlo...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR3 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SQ8ZVTPubMed