BindingDB PrimarySearch

Found 260 of ic50 for UniProtKB: P30559

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50103475(Pmp-Tyr-Ile-Thr-Asn-Cys-Pro-Orn-phe(I,N3)-NH2 | Pm...)copy SMILEScopy InChI

IC50: 0.320nMAssay Description:Ability to inhibit OT-induced inositol phosphate accumulation was determined in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q29S1Q9FPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50100381(5-Oxo-hexanoic acid {1-[((S)-1-carbamoyl-2-thiophe...)copy SMILEScopy InChI

IC50: 1nMAssay Description:Inhibitory concentration required for antagonist activity against oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2T72GQFPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205990(CHEMBL395429 | OXYTOCIN)copy SMILEScopy InChI

IC50: 2.70nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50190528((2R)-2-(2,4-difluorophenyl)-2-[(3R,6R)-3-(2,3-dihy...)copy SMILEScopy InChI

IC50: 3.70nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as inhibition of oxytocin-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q269735QPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50559938(CHEMBL154668)copy SMILES

IC50: 4.60nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2F193D1PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50100380(5-Oxo-hexanoic acid (1-{[(S)-1-carbamoyl-2-(3,4-di...)copy SMILEScopy InChI

IC50: 5nMAssay Description:Inhibitory concentration required for antagonist activity against oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2T72GQFPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410619(CHEMBL2113208)copy SMILEScopy InChI

IC50: 7nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410616(CHEMBL2113185)copy SMILEScopy InChI

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205997(CHEMBL395290 | [Pip7]OT)copy SMILEScopy InChI

IC50: 7nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50027070(CHEMBL2369136)copy SMILEScopy InChI

IC50: 8nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410635(CHEMBL2113211)copy SMILEScopy InChI

IC50: 8nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50384820(EPELSIBAN | GSK557296B)copy SMILEScopy InChI

IC50: 9.20nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516419(CHEMBL4464246)copy SMILEScopy InChI

IC50: 9.30nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516428(CHEMBL4449435)copy SMILEScopy InChI

IC50: 10nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410625(CHEMBL2113201)copy SMILEScopy InChI

IC50: 14nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50326722((Z)-3-(4-(N-(4-chlorophenyl)-N-(2-oxo-2-(2-(2-oxoi...)copy SMILEScopy InChI

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516412(CHEMBL4591825)copy SMILEScopy InChI

IC50: 15nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410634(CHEMBL2113189)copy SMILEScopy InChI

IC50: 15nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50305506(5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5...)copy SMILEScopy InChI

IC50: 23nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516417(CHEMBL4518063)copy SMILEScopy InChI

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205999(CHEMBL434193 | [Mpa1, D-Tyr(Et)2, D-Tic7, D-Tic9]O...)copy SMILEScopy InChI

IC50: 25nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516427(CHEMBL4466263)copy SMILEScopy InChI

IC50: 27nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50178153(4-ethoxy-N-(4-methylphenyl)-N-{2-oxo-2-[2-(2-oxo-1...)copy SMILEScopy InChI

IC50: 30nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516413(CHEMBL4564411)copy SMILEScopy InChI

IC50: 30nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410623(CHEMBL2113179)copy SMILEScopy InChI

IC50: 32nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50459404(CHEMBL4205046)copy SMILEScopy InChI

IC50: 37nMAssay Description:Antagonist activity at OXR receptor (unknown origin)More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205989(CHEMBL393020 | [Mpa1, D-Tyr(Et)2, Pip7]OT)copy SMILEScopy InChI

IC50: 40nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516414(CHEMBL4538696)copy SMILEScopy InChI

IC50: 44nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410621(CHEMBL2113177)copy SMILEScopy InChI

IC50: 49nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205986(CHEMBL233328 | [Mpa1, D-Tyr(Et)2, D-Tic7]OT)copy SMILEScopy InChI

IC50: 51nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516416(CHEMBL4541860)copy SMILEScopy InChI

IC50: 52nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50206001(CHEMBL233080 | [Mpa1, D-Tyr(Et)2, Aib7, D-Tic9]OT)copy SMILEScopy InChI

IC50: 55nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50177595((2S)-5-amino-2-{[(2S)-1-{[(4R,7S,10S,13S,16R)-13-[...)copy SMILEScopy InChI

IC50: 59nMAssay Description:Inhibitory activity against human Oxytocin induced intracellular Calcium mobilization in human Oxytocin receptor transfected HEK293-EBNA cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50410622(CHEMBL2113203)copy SMILEScopy InChI

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BindingDB Entry DOI: 10.7270/Q2QF8TN3PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50305506(5-(3-(3-(2-chloro-4-fluorophenoxy)azetidin-1-yl)-5...)copy SMILEScopy InChI

IC50: 63nMAssay Description:Antagonist activity at human OTR receptor expressed in HEK293FT cells assessed as inhibition of LIT-001-induced response incubated for 30 mins by bet...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50066092(3N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)copy SMILEScopy InChI

IC50: 68nMAssay Description:Antagonistic activity against Oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2D799KHPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50206000(CHEMBL395430 | [Aib7]OT)copy SMILEScopy InChI

IC50: 75nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205987(CHEMBL438849 | [Mpa1, D-Tyr(Et)2, D-Tic7, Aib9]OT)copy SMILEScopy InChI

IC50: 80nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205992(CHEMBL415418 | [Mpa1, L-Tic7]OT)copy SMILEScopy InChI

IC50: 103nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)copy SMILEScopy InChI

IC50: 109nMAssay Description:Antagonist activity at OXR receptor (unknown origin)More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q24J0HRFPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516429(CHEMBL4444840)copy SMILEScopy InChI

IC50: 121nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50133272(CHEMBL406351 | [D-Pen1,Glu4,Lys8]OT)copy SMILEScopy InChI

IC50: 130nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50066084(3N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)copy SMILEScopy InChI

IC50: 130nMAssay Description:Antagonistic activity against Oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2D799KHPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205996(CHEMBL397407 | [L-Tic7]OT)copy SMILEScopy InChI

IC50: 130nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516420(CHEMBL4437214)copy SMILEScopy InChI

IC50: 132nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50133258(CHEMBL2369135 | [D-Pen1,(2S,3R)-p-MeOTMT2,Glu4,Lys...)copy SMILEScopy InChI

IC50: 160nMAssay Description:Binding affinity towards oxytocin receptorMore data for this Ligand-Target Pair

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BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50205995(CHEMBL234377 | [Mpa1, D-Tyr(Et)2, L-Tic7]OT)copy SMILEScopy InChI

IC50: 176nMAssay Description:Displacement of [3H]OT from human OT receptor expressed in HEK cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2P55N5JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516415(CHEMBL4585239)copy SMILEScopy InChI

IC50: 184nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516422(CHEMBL4542267)copy SMILEScopy InChI

IC50: 223nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article
BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Oxytocin receptor(Homo sapiens (Human))
INSERM

Curated by ChEMBL

BDBM50516424(CHEMBL4575160)copy SMILEScopy InChI

IC50: 235nMAssay Description:Antagonist activity at human OTR expressed in HEK293 cells assessed as decrease in calcium flux measured after 10 mins in presence of vasopressin by ...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

PC cid PC sid

Details Article
BindingDB Entry DOI: 10.7270/Q2Q52T0JPubMed

Displayed 1 to 50 (of 260 total ) | Next | Last >>

Targets 1 ▿
- Oxytocin receptor 260
Publications 18 ▿
- ACS Med Chem Lett 10: 996-1001 (2019) 26
- Eur J Med Chem 42: 799-806 (2007) 19
- Eur J Med Chem 143: 1644-1656 (2018) 15
- J Med Chem 48: 7882-905 (2005) 12
- Eur J Med Chem 108: 730-40 (2016) 10
- Eur J Med Chem 136: 330-333 (2017) 9
- J Med Chem 61: 6364-6378 (2018) 7
- J Med Chem 61: 8670-8692 (2018) 7
- Bioorg Med Chem Lett 17: 5796-800 (2007) 6
- J Med Chem 46: 4215-31 (2003) 5
- Bioorg Med Chem Lett 20: 5044-9 (2010) 3
- Bioorg Med Chem Lett 11: 1297-300 (2001) 2
- J Med Chem 41: 3103-27 (1998) 2
- Bioorg Med Chem Lett 21: 1871-5 (2011) 2
- Bioorg Med Chem 26: 3039-3045 (2018) 1
- Bioorg Med Chem Lett 20: 5394-7 (2010) 1
- J Med Chem 44: 3022-30 (2001) 1
- J Med Chem 49: 4159-70 (2006) 1
Institutions 16 ▿
- [The University of Sydney] 34
- [Shanghai Hengrui Pharmaceutical CO., LTD.] 26
- [University of Patras] 19
- [Serono Pharmaceutical Research Institute] 12
- [UMR7200 CNRS/Universit£ de Strasbourg, University of Florida] 7
- [UMR7200 CNRS/Universit£ de Strasbourg, University of Florida] 7
- [Wyeth Research] 6
- [University of Arizona] 5
- [GlaxoSmithKline] 3
- [Merck Research Laboratories, GlaxoSmithKline Medicines Research Centre, MSD] 2
- [Merck Research Laboratories, GlaxoSmithKline Medicines Research Centre, MSD] 2
- [Merck Research Laboratories, GlaxoSmithKline Medicines Research Centre, MSD] 2
- [INSERM, Cardiovascular and Urogenital Centre of Excellence for Drug Discovery, Imperial College, Ligand Pharmaceuticals, Inc.] 1
- [INSERM, Cardiovascular and Urogenital Centre of Excellence for Drug Discovery, Imperial College, Ligand Pharmaceuticals, Inc.] 1
- [INSERM, Cardiovascular and Urogenital Centre of Excellence for Drug Discovery, Imperial College, Ligand Pharmaceuticals, Inc.] 1
- [INSERM, Cardiovascular and Urogenital Centre of Excellence for Drug Discovery, Imperial College, Ligand Pharmaceuticals, Inc.] 1
Affinity: 0.32 to 1.0E+5 nM▿
- IC50 260
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 11