Compile Data Set for Download or QSAR
Found 78 of ic50 for UniProtKB: P9WKE1
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498068(CHEMBL3394234)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498069(CHEMBL3394233)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498093(CHEMBL3394236)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498070(CHEMBL3394163)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498082(CHEMBL3394237)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498096(CHEMBL3394232)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498089(CHEMBL3394162)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498090(CHEMBL3394161)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498057(CHEMBL3394235)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498060(CHEMBL3394249)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498059(CHEMBL3394250)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498061(CHEMBL3394247)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574965(CHEMBL4876372)copy SMILES
Affinity DataIC50: 120nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574967(CHEMBL4858644)copy SMILES
Affinity DataIC50: 140nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498062(CHEMBL3394246)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498056(CHEMBL3394242)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574975(CHEMBL4869914)copy SMILES
Affinity DataIC50: 220nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498080(CHEMBL3394245)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498074(CHEMBL3394155)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498079(CHEMBL3394248)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498088(CHEMBL3394240)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498085(CHEMBL3394151)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498073(CHEMBL3394157)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574970(CHEMBL4860538)copy SMILES
Affinity DataIC50: 450nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574963(CHEMBL4848605)copy SMILES
Affinity DataIC50: 600nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574972(CHEMBL4876370)copy SMILES
Affinity DataIC50: 600nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574964(CHEMBL4868830)copy SMILES
Affinity DataIC50: 650nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574973(CHEMBL4874579)copy SMILES
Affinity DataIC50: 770nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574974(CHEMBL4865732)copy SMILES
Affinity DataIC50: 810nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498063(CHEMBL3394244)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574956(CHEMBL4854974)copy SMILES
Affinity DataIC50: 890nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498065(CHEMBL3394241)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498058(CHEMBL3394153)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574955(CHEMBL4860579)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574961(CHEMBL4854518)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574968(CHEMBL4871611)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574960(CHEMBL4849731)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498094(CHEMBL3394154)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498091(CHEMBL3394160)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498077(CHEMBL3394148)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498054(CHEMBL1477426)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498078(CHEMBL3394146)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498064(CHEMBL3394243)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574943(CHEMBL4870416)copy SMILES
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574962(CHEMBL4863370)copy SMILES
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498084(CHEMBL3394156)copy SMILEScopy InChI
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50498095(CHEMBL3394152)copy SMILEScopy InChI
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis thymidylate kinase activity by pyruvate kinase-lactate dehydrogenase coupled assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9TD7PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574971(CHEMBL4868671)copy SMILES
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574966(CHEMBL4855593)copy SMILES
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50574958(CHEMBL4846640)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv TMPK expressed in Escherichia coli by coupled enzyme based spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BM5PubMed
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