Compile Data Set for Download or QSAR
Found 14 of ic50 for UniProtKB: P58406
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328807((2R,4S,5S)-1,2,5-trimethyl-4-(2-(naphthalen-1-yl)e...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328802((2R,4S,5S)-1,2,5-trimethyl-4-(naphthalen-1-ylethyn...)copy SMILEScopy InChI
Affinity DataIC50: 119nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328809(CHEMBL1270165 | rac-1,2,5-trimethyl-4-(2-(naphthal...)copy SMILEScopy InChI
Affinity DataIC50: 122nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328801(1,2,5-trimethyl-4-(naphthalen-1-ylethynyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328810(CHEMBL1270166 | rac-6-methyl-7-(naphthalen-1-yleth...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328811(CHEMBL1270167 | rac-6-methyl-7-(2-(naphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 345nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328806(CHEMBL1270058 | rac-1,2,5-trimethyl-4-(2-(naphthal...)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328805(CHEMBL1269952 | rac-1,2,5-trimethyl-4-(2-(naphthal...)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328812(CHEMBL1270264 | rac-1,2,5-trimethyl-4-(quinolin-5-...)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328808(CHEMBL1270060 | rac-1,2,5-trimethyl-4-(naphthalen-...)copy SMILEScopy InChI
Affinity DataIC50: 810nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328803((2S,4R,5R)-1,2,5-trimethyl-4-(naphthalen-1-ylethyn...)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328813(CHEMBL1270265 | rac-1,2,5-trimethyl-4-(quinolin-8-...)copy SMILEScopy InChI
Affinity DataIC50: 9.73E+3nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys Inc.

Curated by ChEMBL
LigandPNGBDBM50328804(CHEMBL1269951 | rac-1,2,5-trimethyl-4-(naphthalen-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6RGGPubMed