Compile Data Set for Download or QSAR
Found 24 of ic50 for UniProtKB: P97571
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50114340((S)-2-(4-Fluoro-benzenesulfonylamino)-N-((S)-1-for...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358131(CHEMBL1923954)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358138(CHEMBL1923961)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358132(CHEMBL1923955)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358137(CHEMBL1923960)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358140(CHEMBL1923963)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358134(CHEMBL1923957)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358133(CHEMBL1923956)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358139(CHEMBL1923962)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358136(CHEMBL1923959)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358142(CHEMBL1923965)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358143(CHEMBL1923966)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258383(CHEMBL4063636)copy SMILEScopy InChI
Affinity DataIC50: 591nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358135(CHEMBL1923958)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358141(CHEMBL1923964)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258312(CHEMBL4095528)copy SMILEScopy InChI
Affinity DataIC50: 971nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258392(CHEMBL4092996)copy SMILEScopy InChI
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258317(CHEMBL4072233)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258313(CHEMBL4104445)copy SMILEScopy InChI
Affinity DataIC50: 5.18E+3nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50258316(CHEMBL4094544)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of calpain-1 in rat hippocampal slices assessed as prevention of NMDA-induced spectrin cleavage preincubated for 30 mins followed by NMDA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242P4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50124010(2-(4-Fluoro-benzenesulfonylamino)-N-(1-formyl-3-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358144(CHEMBL1923967)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358145(CHEMBL1923968)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed
TargetCalpain-1 catalytic subunit(Rattus norvegicus)
University of Canterbury

Curated by ChEMBL
LigandPNGBDBM50358146(CHEMBL1923969)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat CAPN1 using BODIPY-labeled casein substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PJ4PubMed