Compile Data Set for Download or QSAR
Found 33 of ic50 for UniProtKB: P27008
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276150(2-(2,2,6,6-Tetramethyl-1,2,3,6-tetrahydropyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276874(2-(1-Oxyl-2,2,6,6-tetramethyl-1,2,3,6-tetrahydropy...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276945(2-(1,2,2,5,5-pentamethyl-2,5-dihydro-1H-pyrrol-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276946(2-(1-Acetyl-2,2,5,5-pentamethyl-2,5-dihydro-1H-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276947(2-(1-Methoxy-2,2,5,5-pentamethyl-2,5-dihydro-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276872(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276148(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276112(2-[4-(3-Trifluoromethylphenyl)-2,2,5,5-tetramethyl...)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276110(2-(4-Bromo-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 137nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276201(2-[1-Oxyl-4-(3-trifluoromethylphenyl)-2,2,5,5-tetr...)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276199(2-(4-Bromo-1-oxyl-2,2,5,5-tetramethyl-2,5-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 201nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276109(4-(4-Carbamoyl-1H-benzimidazol-2-yl)-2,2,5,5-tetra...)copy SMILEScopy InChI
Affinity DataIC50: 216nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276111(2-(4-Phenyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276108(2-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 345nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276203(2-(4,4,6,6-Tetramethyl-5,6-dihydro-4H-thieno[3,4-c...)copy SMILEScopy InChI
Affinity DataIC50: 354nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276202(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)copy SMILEScopy InChI
Affinity DataIC50: 432nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276204(2-(1,1,3,3-Tetramethyl-2,3-dihydro-1H-isoindol-5-y...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276205(2-(1,1,3,3-Tetramethyl-2,3-dihydro-1H-pyrrolo[3,4-...)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276943(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 472nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276875(2-[4-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 564nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276151(2-[4-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-...)copy SMILEScopy InChI
Affinity DataIC50: 572nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276197(2-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 721nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276200(2-(1-Oxyl-4-phenyl-2,2,5,5-tetramethyl-2,5-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276873(2-[4-Dibenzofuran-4-yl-1-oxyl-2,2,5,5-tetramethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276149(2-[4-Dibenzofuran-4-yl-2,2,5,5-tetramethyl-2,5-dih...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276114(2-((2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrrol-3-yl...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276944(2-(5-Oxyl-4,4,6,6-tetramethyl-5,6-dihydro-4H-thien...)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276113(2-((2,2,6,6-tetramethyl-1,2,3,6-tetrahydropyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50413274(CHEMBL2094004)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50413275(CHEMBL2094005)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276116(2-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276115(1-(1-Oxyl-2,2,5,5-tetramethyl-2,5-dihydro-1H-pyrro...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed
TargetPoly [ADP-ribose] polymerase 1(Rattus norvegicus)
University of Pecs

Curated by ChEMBL
LigandPNGBDBM50276152(2-(2,2,5,5-Tetramethyl-2,5-dihydro-1H-pyrrol-3-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat liver PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29S1QXHPubMed