Compile Data Set for Download or QSAR
Found 5 of ic50 for UniProtKB: P18493
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)TBA
LigandPNGBDBM27709(2-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin...)copy SMILEScopy InChI
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)TBA
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of calf thymus PARP1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M65KBPubMed
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)TBA
LigandPNGBDBM27503(5-AIQ | 5-amino-1,2-dihydroisoquinolin-1-one | 5-a...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of calf thymus PARP-1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BP047DPubMed
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)TBA
LigandPNGBDBM27500(5,6-dihydrophenanthridin-6-one | 5H-Phenanthridin-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of calf thymus ARTD1 assessed as incorporation of [Ade-U-14C]-NAD+ after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB477RPubMed
TargetPoly [ADP-ribose] polymerase 1(Bos taurus)TBA
LigandPNGBDBM50446131(CHEMBL3108871)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:Inhibition of bovine ARTD1 assessed as incorporation of [adenine-2,8-3H]NAD after 1 hr by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SB477RPubMed