Compile Data Set for Download or QSAR
Found 12 of ic50 for UniProtKB: P49185
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50373215(CHEMBL259060)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced AP1 phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JS9R8MPubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376114(CHEMBL259720)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376124(CHEMBL261413)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376125(CHEMBL411083)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376112(CHEMBL258845)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376111(CHEMBL258618)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376123(CHEMBL260064)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376122(CHEMBL260065)copy SMILEScopy InChI
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376110(CHEMBL409350)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376115(CHEMBL437107)copy SMILEScopy InChI
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50376120(CHEMBL259554)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 8(Rattus norvegicus)
Takeda Pharmaceutical Company, Ltd

Curated by ChEMBL
LigandPNGBDBM50373215(CHEMBL259060)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of JNK1 in rat H9c2 cells assessed as inhibition of anisomycin-induced cJun phosphorylation after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP2598PubMed