Compile Data Set for Download or QSAR
Found 4 of ic50 for UniProtKB: P70658
TargetC-X-C chemokine receptor type 4(Mus musculus)
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50326057(([5-(4-Methyl-1-piperazinyl)-2-({methyl[(8S)-5,6,7...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at mouse CXCR4 expressed in human U2OS cells assessed as inhibition of SDF1-induced increase in intracellular calcium level by FL...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47PBFPubMed
TargetC-X-C chemokine receptor type 4(Mus musculus)
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50270016(CHEMBL4070320)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Antagonist activity at mouse CXCR4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QTHPubMed
TargetC-X-C chemokine receptor type 4(Mus musculus)
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50270018(CHEMBL4075205)copy SMILEScopy InChI
Affinity DataIC50: 9.20nMAssay Description:Antagonist activity at mouse CXCR4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QTHPubMed
TargetC-X-C chemokine receptor type 4(Mus musculus)
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50270019(CHEMBL4065224)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at mouse CXCR4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QTHPubMed