Compile Data Set for Download or QSAR
Found 16 of ic50 for UniProtKB: P53610
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat brain GGTase1 assessed as decrease in transfer of [3H]H]geranylgeranyl from [3H]geranylgeranyl PPi to H-Ras-CVLL after 30 mins by l...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542R5NPubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481906(CHEMBL1075839)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481911(CHEMBL1075809)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481907(CHEMBL1075810)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481909(CHEMBL1075863)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481908(CHEMBL1075861)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481912(CHEMBL1075865)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50481910(CHEMBL1075859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat recombinant GGTase-1 by SDS-PAGE end point assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CS3PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504717(CHEMBL4459281)copy SMILEScopy InChI
Affinity DataIC50: 1.22E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504718(CHEMBL4564870)copy SMILEScopy InChI
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50273716(CHEMBL457423 | [2-(Benzoimidazol-1-yl)ethyl]-bisph...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504719(CHEMBL4438314)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504720(CHEMBL4529809)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504715(CHEMBL4514446)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504714(CHEMBL4460301)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed
TargetGeranylgeranyl transferase type-1 subunit beta(Rattus norvegicus)
Temple University

Curated by ChEMBL
LigandPNGBDBM50504716(CHEMBL4589567)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of recombinant rat GGtase-1 expressed in Escherichia coli using dansyl-GCVLL as substrate after 1.5 hrs by spectrofluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2DW5PubMed