Compile Data Set for Download or QSAR
Found 3 of ic50 for UniProtKB: P10499
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237249(CHEMBL4076021)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)4 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed