Compile Data Set for Download or QSAR
Found 45 of ic50 for UniProtKB: P9WFV1
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241780(CHEMBL4105269)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241754(CHEMBL4077894)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Binding affinity against sigma receptor from guinea pig brain, using [3H](+)-3-PPP as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241778(CHEMBL4086672)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241756(CHEMBL4075879)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241795(CHEMBL4104309)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241792(CHEMBL4102148)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241791(CHEMBL4082544)copy SMILEScopy InChI
Affinity DataIC50: 92nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241781(CHEMBL4066833)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241782(CHEMBL4081207)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241755(CHEMBL4081755)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Binding affinity against sigma receptor from guinea pig brain, using [3H](+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241789(CHEMBL4084478)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241757(CHEMBL4066786)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241772(CHEMBL4105458)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241769(CHEMBL4090012)copy SMILEScopy InChI
Affinity DataIC50: 160nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241760(CHEMBL4067937)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)copy SMILEScopy InChI
Affinity DataIC50: 216nMAssay Description:Inhibition of Mycobacterium tuberculosis LeuRS expressed in Escherichia coli Rosetta (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z480DPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241798(CHEMBL4084509)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241759(CHEMBL4094412)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241770(CHEMBL4061966)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241800(CHEMBL4074178)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241799(CHEMBL4096785)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241766(CHEMBL4087944)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241775(CHEMBL4078760)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241793(CHEMBL4066921)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241767(CHEMBL4076333)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241758(CHEMBL4104573)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241794(CHEMBL4075254)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241761(CHEMBL4089141)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Binding affinity against sigma receptor from guinea pig brain, using [3H](+)-pentazocine as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241783(CHEMBL4081973)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241776(CHEMBL4071439)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241777(CHEMBL4092224)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241763(CHEMBL4103410)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241765(CHEMBL4080074)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241768(CHEMBL4062832)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241788(CHEMBL4062801)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241774(CHEMBL4070589)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241762(CHEMBL4087629)copy SMILEScopy InChI
Affinity DataIC50: 690nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241764(CHEMBL4065024)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241787(CHEMBL4100936)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241786(CHEMBL4099978)copy SMILEScopy InChI
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241801(CHEMBL4077080)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241771(CHEMBL4100159)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241790(CHEMBL4081018)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals, Inc.

Curated by ChEMBL
LigandPNGBDBM50241773(CHEMBL4097736)copy SMILEScopy InChI
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD13THPubMed