Compile Data Set for Download or QSAR
Found 78 of ic50 for UniProtKB: P28347
LigandPNGBDBM626350(2-[[[4-cyano-7-(4-isopropyl-2- thienyl)-2,3-dihyd...)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626331(US11787775, Compound 16-C)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626318(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50271260(CHEMBL4130196)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human His-tagged YAP (50 to 171 residues) interaction with human GST-tagged TEAD1 (194 to 411) expressed in Escherichia coli BL21(DE3) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91H7PubMed
LigandPNGBDBM50497300(CHEMBL3335461)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626361(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)copy SMILES
Affinity DataIC50: 30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626333(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)copy SMILES
Affinity DataIC50: 30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)copy SMILES
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497290(CHEMBL3335458)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM50497304(CHEMBL3335453)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626334(2-[[[4-cyano-7-[4-(1,1- difluoroethyl)phenyl]-2,3...)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626342(2-[[[4-cyano-7-(2-fluoro-4- isopropyl-phenyl)-2,3...)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626354(2-[[[4-cyano-2,2-dideuterio-7-[4- (trifluorometho...)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626330(2-[[[4-cyano-7-[4- (trifluoromethyl)phenyl]-2,3- ...)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626362(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626324(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626336(2-[[[4-fluoro-7-(4-isopropylphenyl)- 2,3-dihydrob...)copy SMILES
Affinity DataIC50: 60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626323(US11787775, Compound 8 | methyl 2-[[[4-cyano-7-(4-...)copy SMILES
Affinity DataIC50: 70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497306(CHEMBL3335463)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626332(US11787775, Compound 16-D)copy SMILES
Affinity DataIC50: 80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626358(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)copy SMILES
Affinity DataIC50: 80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50271259(CHEMBL4129172)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of Gal4-fused TEAD 1 (unknown origin) interaction with YAP expressed in human 293T cells by Dual-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B91H7PubMed
LigandPNGBDBM626337(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrofu...)copy SMILES
Affinity DataIC50: 90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626355(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)copy SMILES
Affinity DataIC50: 90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626360(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)copy SMILES
Affinity DataIC50: 110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497296(CHEMBL3335452)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626338(2-[[[7-cyano-4-[4-(1,1- difluoroethyl)phenyl]-1,3...)copy SMILES
Affinity DataIC50: 160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626352(2-[[[4-(hydroxymethyl)-7-[4- (trifluoromethoxy)ph...)copy SMILES
Affinity DataIC50: 160nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626319(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626326(7-(4-isopropylphenyl)-5-[(2- methylene-3-oxo-buty...)copy SMILES
Affinity DataIC50: 180nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626335(2-[[[4-(4-isopropylphenyl)-6,7- dihydrofuro[3,2-d...)copy SMILES
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626365(2-[[[7-cyano-4-[4-(pentafluoro- lambda6-sulfanyl)...)copy SMILES
Affinity DataIC50: 200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626316(2-[[[7-(4-isopropylphenyl)-2,3- dihydrobenzofuran...)copy SMILES
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626363(2-[[[4-cyano-7-[4-(pentafluoro- lambda6-sulfanyl)...)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626324(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626347(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)copy SMILES
Affinity DataIC50: 310nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497288(CHEMBL3335456)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626364(2-[[[4-cyano-7-(5-isopropylthiazol- 2-yl)-2,3-dih...)copy SMILES
Affinity DataIC50: 310nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626319(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 320nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497308(CHEMBL3335457)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM50497297(CHEMBL3335459)copy SMILEScopy InChI
Affinity DataIC50: 350nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM50497289(CHEMBL3335454)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626344(2-[[[7-cyano-4-[4- (trifluoromethoxy)phenyl]-1,3-...)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497302(CHEMBL3335460)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626359(2-[[[4-cyano-7-[4- (trifluoromethoxy)phenyl]-2,3-...)copy SMILES
Affinity DataIC50: 400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626329(2-[[[4-(hydroxymethyl)-7-(4- isopropylphenyl)-2,3...)copy SMILES
Affinity DataIC50: 520nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50497309(CHEMBL3335462)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of YAP/ GST-TEAD1 (unknown origin) interaction by surface plasmon resonance assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63H7PubMed
LigandPNGBDBM626322(2-[[[4-cyano-7-(4-isopropylphenyl)- 2,3-dihydrobe...)copy SMILES
Affinity DataIC50: 540nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM626339(2-[[[6-methoxy-5-[(E)-2-[trans-4- (trifluoromethy...)copy SMILES
Affinity DataIC50: 580nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
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