Compile Data Set for Download or QSAR
Found 25 of ic50 for UniProtKB: P56719
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97406(Orexin receptor antagonist 1 | US20130102619, 1)copy SMILEScopy InChI
Affinity DataIC50: 12nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97397(Orexin receptor antagonist 29 | Orexin receptor an...)copy SMILEScopy InChI
Affinity DataIC50: 12nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97397(Orexin receptor antagonist 29 | Orexin receptor an...)copy SMILEScopy InChI
Affinity DataIC50: 17nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97373(Orexin receptor antagonist 5 | US20130102619, 5)copy SMILEScopy InChI
Affinity DataIC50: 17nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97408(Orexin receptor antagonist 3 | US20130102619, 3)copy SMILEScopy InChI
Affinity DataIC50: 18nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97375(Orexin receptor antagonist 6 | US20130102619, 6)copy SMILEScopy InChI
Affinity DataIC50: 18nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97378(Orexin receptor antagonist 9 | US20130102619, 9)copy SMILEScopy InChI
Affinity DataIC50: 22nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97390(Orexin receptor antagonist 22 | US20130102619, 22)copy SMILEScopy InChI
Affinity DataIC50: 23nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97407(Orexin receptor antagonist 2 | US20130102619, 2)copy SMILEScopy InChI
Affinity DataIC50: 28nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97377(Orexin receptor antagonist 8 | US20130102619, 8)copy SMILEScopy InChI
Affinity DataIC50: 29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97379(Orexin receptor antagonist 10 | US20130102619, 10)copy SMILEScopy InChI
Affinity DataIC50: 29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97374(Orexin receptor antagonist 4 | US20130102619, 4)copy SMILEScopy InChI
Affinity DataIC50: 29nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97403(Orexin receptor antagonist 35 | US20130102619, 35)copy SMILEScopy InChI
Affinity DataIC50: 31nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97399(Orexin receptor antagonist 31 | US20130102619, 31)copy SMILEScopy InChI
Affinity DataIC50: 38nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97400(Orexin receptor antagonist 32 | US20130102619, 32)copy SMILEScopy InChI
Affinity DataIC50: 44nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97404(Orexin receptor antagonist 36 | US20130102619, 36)copy SMILEScopy InChI
Affinity DataIC50: 47nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97402(Orexin receptor antagonist 34 | US20130102619, 34)copy SMILEScopy InChI
Affinity DataIC50: 48nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97401(Orexin receptor antagonist 33 | US20130102619, 33)copy SMILEScopy InChI
Affinity DataIC50: 52nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97384(Orexin receptor antagonist 15 | US20130102619, 15)copy SMILEScopy InChI
Affinity DataIC50: 62nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97383(Orexin receptor antagonist 14 | US20130102619, 14)copy SMILEScopy InChI
Affinity DataIC50: 65nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97388(Orexin receptor antagonist 20 | US20130102619, 20)copy SMILEScopy InChI
Affinity DataIC50: 67nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97385(Orexin receptor antagonist 17 | US20130102619, 17)copy SMILEScopy InChI
Affinity DataIC50: 82nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM97398(Orexin receptor antagonist 30 | US20130102619, 30)copy SMILEScopy InChI
Affinity DataIC50: 110nMT: 2°CAssay Description:FLIPR assay using orexin receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K64GP7US Patent
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM50060937(CHEMBL3394848)copy SMILEScopy InChI
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at rat OX2 receptor assessed as inhibition of Ala-6,12 orexin-A-induced calcium increase preincubated for 5 mins prior to Ala-6,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VRGPubMed
TargetOrexin receptor type 2(Rattus norvegicus (Rat))
TBA

US Patent
LigandPNGBDBM50203731(CHEMBL3973097)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at rat OX2 receptor assessed as inhibition of Ala-6,12 orexin-A-induced calcium increase preincubated for 5 mins prior to Ala-6,1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VRGPubMed