Compile Data Set for Download or QSAR
Found 31 of ic50 for UniProtKB: P51531
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394585(2-(6-amino-5-(1-(1- | US10308614, Example 188)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394575(2-(6-amino-5-(2- | US10308614, Example 178)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394605(2-(6-amino-5-cyclohexylpyridazin-3-yl)phenol | US1...)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394584(2-(6-amino-5-(1-methyl- | US10308614, Example 187)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394567((S)-2-(6-amino-5-(1- | US10308614, Example 170)copy SMILEScopy InChI
Affinity DataIC50: 14.9nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394528(1-(4-(3-amino-6-(2- | US10308614, Example 129)copy SMILEScopy InChI
Affinity DataIC50: 18.4nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394571(2-(6-amino-5- | US10308614, Example 174)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394403(2-(6-amino-5-(4-((dimethylami- | US10308614, Examp...)copy SMILEScopy InChI
Affinity DataIC50: 22.5nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394606(2-(6-amino-5- | US10308614, Example 210)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394456(2-(6-amino-5-(3- | US10308614, Example 57)copy SMILEScopy InChI
Affinity DataIC50: 35.6nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394507(2-(6-amino-5-(3-methyl-4-(methylsulfonyl)piperazin...)copy SMILEScopy InChI
Affinity DataIC50: 35.8nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394414(2-(6-amino-5-(4-(1- | US10308614, Example 15)copy SMILEScopy InChI
Affinity DataIC50: 36.1nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394583(2-(6-amino-5-phenylpyridazin-3-yl)phenol | US10308...)copy SMILEScopy InChI
Affinity DataIC50: 37.3nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394521(1-(4-(3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl)-2...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394614(2-(6-amino-5-(1-benzylpiperidin-4-yl)pyridazin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 39.3nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394490(2-(6-amino-5-(piperidin-1-yl)pyridazin-3-yl)phenol...)copy SMILEScopy InChI
Affinity DataIC50: 45.9nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394518(2-(6-amino-5-(3-benzyl- | US10308614, Example 119)copy SMILEScopy InChI
Affinity DataIC50: 46.8nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394408(2-(6-amino-5-((3aR,6aS)-5- | US10308614, Example 9)copy SMILEScopy InChI
Affinity DataIC50: 47.6nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394586(2-(6-amino-5-(4- | US10308614, Example 189)copy SMILEScopy InChI
Affinity DataIC50: 49.3nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394577(2-(6-amino-5-((1- | US10308614, Example 180)copy SMILEScopy InChI
Affinity DataIC50: 59.7nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394401(2-(6-amino-5-(4-(pyridin- | US10308614, Example 3)copy SMILEScopy InChI
Affinity DataIC50: 60.7nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394432(2-(6-amino-5-(2,6- | US10308614, Example 33)copy SMILEScopy InChI
Affinity DataIC50: 69.6nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394444(2-(6-amino-5- | US10308614, Example 45)copy SMILEScopy InChI
Affinity DataIC50: 71.5nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394402(1-(4-(3-amino-6-(2- | US10308614, Example 4)copy SMILEScopy InChI
Affinity DataIC50: 71.7nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394415(2-(6-amino-5-(8-benzyl-3,8- | US10308614, Example ...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394574(2-(6-amino-5-((1- | US10308614, Example 177)copy SMILEScopy InChI
Affinity DataIC50: 92.5nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394565(2-(6-amino-5-(1- | US10308614, Example 168)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394570(2-(6-amino-5-(2- | US10308614, Example 173)copy SMILEScopy InChI
Affinity DataIC50: 276nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394602(2-(6-amino-5-phenylpyridazin-3-yl)-6-fluorophenol ...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394613(2-(6-amino-5-(1-(phenylsulfonyl)pyrrolidin-3-yl)py...)copy SMILEScopy InChI
Affinity DataIC50: 466nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent
TargetIsoform Short of Probable global transcription activator SNF2L2 (Short) 377-1486](Homo sapiens (Human))
The Institute of Cancer Research

LigandPNGBDBM394600(2-(6-(methylamino)pyridazin-3-yl)phenol | US103086...)copy SMILEScopy InChI
Affinity DataIC50: 1.04E+3nMAssay Description:Histidine epitope tagged BRM (Isoform 2) Bromodomain1377-1486 (S1377-Q1486; Swiss Prot P51531-2; mhhhhhhgslvpr\gsSPNPPKLTKQMNAIIDTVINYKDSSGRQLSEVFIQL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26112NJUS Patent