Compile Data Set for Download or QSAR
Found 30 of ki for UniProtKB: P49768
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50575178(CHEMBL4853450)copy SMILES
Affinity DataKi:  0.420nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HGFPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50575197(CHEMBL4868549)copy SMILES
Affinity DataKi:  0.650nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HGFPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476859(CHEMBL232938)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476878(CHEMBL399204)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476861(CHEMBL401044)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50575187(CHEMBL4848116)copy SMILES
Affinity DataKi:  1.20nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HGFPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476880(CHEMBL450279)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476871(CHEMBL232182)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476864(CHEMBL429438)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476860(CHEMBL232936)copy SMILEScopy InChI
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476870(CHEMBL232346)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50575179(CHEMBL4851959)copy SMILES
Affinity DataKi:  2.60nMAssay Description:Noncompetitive inhibition of gamma secretase (unknown origin) expressed in HEK293 cells assessed as reduction of A-beta40 levels using varying level ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1HGFPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM209909(US9273014, Comparative Compound 45 | US9427442, Co...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476872(CHEMBL401045)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476865(CHEMBL392265)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476857(CHEMBL449960)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476862(CHEMBL232739)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476856(CHEMBL232138)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476866(CHEMBL231941)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476875(CHEMBL232183)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476879(CHEMBL233172)copy SMILEScopy InChI
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476873(CHEMBL231984)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476858(CHEMBL231725)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476876(CHEMBL399819)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476868(CHEMBL232367)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476869(CHEMBL232968)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476874(CHEMBL393520)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476863(CHEMBL273493)copy SMILEScopy InChI
Affinity DataKi:  111nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476877(CHEMBL398379)copy SMILEScopy InChI
Affinity DataKi:  227nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed
TargetPresenilin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50476867(CHEMBL401434)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]succinamide from gamma secretase in THP1 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90CFPPubMed