Compile Data Set for Download or QSAR
Found 21 of ki for UniProtKB: P06869
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531924(CHEMBL4464577)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499240(CHEMBL3735080)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531926(CHEMBL4550668)copy SMILEScopy InChI
Affinity DataKi:  246nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)copy SMILEScopy InChI
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)copy SMILEScopy InChI
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499239(CHEMBL3734777)copy SMILEScopy InChI
Affinity DataKi:  550nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50529264(CHEMBL4513418)copy SMILEScopy InChI
Affinity DataKi:  956nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639TNCPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459059(CHEMBL4217043)copy SMILEScopy InChI
Affinity DataKi:  1.61E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50531925(CHEMBL4522772)copy SMILEScopy InChI
Affinity DataKi:  1.77E+3nMAssay Description:Inhibition of mouse uPA serine protease domain preincubated for 15 mins followed by chromogenic substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1V6RPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459054(CHEMBL4213248)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)copy SMILEScopy InChI
Affinity DataKi:  2.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459080(CHEMBL4211423)copy SMILEScopy InChI
Affinity DataKi:  2.77E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639TNCPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50459079(CHEMBL4206764)copy SMILEScopy InChI
Affinity DataKi:  3.29E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2639TNCPubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM81818(CAS_1794 | CHEMBL1909810 | HMA | NSC_1794)copy SMILEScopy InChI
Affinity DataKi:  9.31E+3nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WH4PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499238(CHEMBL3735263)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499242(CHEMBL3736473)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499241(CHEMBL3735513)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed
TargetUrokinase-type plasminogen activator(Mus musculus (Mouse))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50499237(CHEMBL3735217)copy SMILEScopy InChI
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of mouse uPA for 15 mins using pyro-Glu-Gly-Arg-p-nitroanilide as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8JH7PubMed