TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Irreversible inhibition of human FGFR3 preincubated with enzyme followed by peptide substrate addition by caliper capillary electrophoresis methodMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.31nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.31nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.51nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.51nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.51nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.51nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.65nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.65nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.78nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.78nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.93nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 6.93nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.06nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.16nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.16nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.16nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.16nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.35nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.35nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.42nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.68nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.78nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.78nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.07nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.07nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.14nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.32nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.47nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.47nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.65nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.85nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 8.96nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.04nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.04nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.31nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.31nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.39nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.42nMAssay Description:The inhibitory activities of compounds of the invention against FGFR3 (FGFR3 Kinase Enzyme System: Promega), were evaluated by mixing the FGFR3 prote...More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Principia Biopharma, Inc.
Curated by ChEMBL
Principia Biopharma, Inc.
Curated by ChEMBL
Affinity DataKi: 9.42nMAssay Description:Assay was performed in buffer containing 40 mM Tris pH 7.5, 20 mM MgCl2, 0.1 mg/mL BSA, 1 mM DTT and 2 mM MnCl2. The inhibitory activities of compoun...More data for this Ligand-Target Pair
