Compile Data Set for Download or QSAR
Found 29 of kd for UniProtKB: P54619
LigandPNGBDBM237920(US9394285, 1)copy SMILEScopy InChI
Affinity DataKd:  9nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
LigandPNGBDBM237920(US9394285, 1)copy SMILEScopy InChI
Affinity DataKd:  9nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
LigandPNGBDBM237920(US9394285, 1)copy SMILEScopy InChI
Affinity DataKd:  9nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
LigandPNGBDBM50505541(CHEMBL4465866)copy SMILEScopy InChI
Affinity DataKd:  13nMAssay Description:Binding affinity to recombinant human full-length GST N-Terminal tagged-AMPK alpha1/N-Terminal GST tagged-AMPK beta1/N-Terminal his-tagged AMPK gamma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S0KPubMed
LigandPNGBDBM238084(US9394285, 178 | US9394285, 179)copy SMILES
Affinity DataKd:  14nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM50244667(CHEMBL4105032)copy SMILEScopy InChI
Affinity DataKd:  14nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM50244667(CHEMBL4105032)copy SMILEScopy InChI
Affinity DataKd:  14nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q242WTPubMed
LigandPNGBDBM238079(US9394285, 173)copy SMILEScopy InChI
Affinity DataKd:  14nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
LigandPNGBDBM238079(US9394285, 173)copy SMILEScopy InChI
Affinity DataKd:  14nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
LigandPNGBDBM50505542(CHEMBL4576489)copy SMILEScopy InChI
Affinity DataKd:  15nMAssay Description:Binding affinity to recombinant human full-length GST N-Terminal tagged-AMPK alpha1/N-Terminal GST tagged-AMPK beta1/N-Terminal his-tagged AMPK gamma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0S0KPubMed
LigandPNGBDBM237925(US9394285, 6)copy SMILEScopy InChI
Affinity DataKd:  20nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM237958(US9394285, 39)copy SMILEScopy InChI
Affinity DataKd:  22nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM237984(US9394285, 67)copy SMILEScopy InChI
Affinity DataKd:  23nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BRCPubMed
LigandPNGBDBM237923(US9394285, 4)copy SMILEScopy InChI
Affinity DataKd:  48nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM237931(US9394285, 12)copy SMILEScopy InChI
Affinity DataKd:  48nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM50195537(CHEMBL3957427)copy SMILEScopy InChI
Affinity DataKd:  74nMAssay Description:Binding affinity for full length human N-terminal His/BAP-tagged AMPK alpha1/beta1/gamma1 expressed in Escherichia coli BL21-CodonPlus by surface pla...More data for this Ligand-Target Pair
LigandPNGBDBM237952(US9394285, 33)copy SMILEScopy InChI
Affinity DataKd:  90nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BRCPubMed
LigandPNGBDBM50463100(CHEMBL4249790)copy SMILEScopy InChI
Affinity DataKd:  113nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
LigandPNGBDBM237921(US9394285, 2)copy SMILEScopy InChI
Affinity DataKd:  150nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BRCPubMed
LigandPNGBDBM50463099(CHEMBL4246000)copy SMILEScopy InChI
Affinity DataKd:  198nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
LigandPNGBDBM50463101(CHEMBL4250253)copy SMILEScopy InChI
Affinity DataKd:  209nMAssay Description:Binding affinity to Bap-tagged human AMPKalpha1beta1gamma1 expressed in Escherichia coli BL21 cells by SPR analysisMore data for this Ligand-Target Pair
LigandPNGBDBM50244665(CHEMBL4097332)copy SMILEScopy InChI
Affinity DataKd:  410nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM50242401(4-hydroxy-3-(2'-hydroxybiphenyl-4-yl)-6-oxo-6,7-di...)copy SMILEScopy InChI
Affinity DataKd:  487nMAssay Description:Binding affinity for full length human N-terminal His/BAP-tagged AMPK alpha1/beta1/gamma1 expressed in Escherichia coli BL21-CodonPlus by surface pla...More data for this Ligand-Target Pair
LigandPNGBDBM50242401(4-hydroxy-3-(2'-hydroxybiphenyl-4-yl)-6-oxo-6,7-di...)copy SMILEScopy InChI
Affinity DataKd:  510nMAssay Description:Binding affinity to human recombinant N-terminal AVI-tagged phosphorylated AMPK alpha1beta1gamma1 expressed in Escherichia coli BL21 cells after 1 to...More data for this Ligand-Target Pair
LigandPNGBDBM50244669(CHEMBL4079303)copy SMILEScopy InChI
Affinity DataKd:  580nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM50244636(CHEMBL4087189)copy SMILEScopy InChI
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human BAP-tagged AMPK alpha1/beta1/gamma1 by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028TZTPubMed
LigandPNGBDBM60978(6-Chloro-5-(4-methoxyphenyl)-1H-indazole-3-carboxy...)copy SMILEScopy InChI
Affinity DataKd:  1.78E+3nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BRCPubMed
LigandPNGBDBM18137(AMP | CHEMBL752 | US11185100, TABLE 7.3 | [(2R,3S,...)copy SMILEScopy InChI
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
LigandPNGBDBM50191352(CHEMBL3936376)copy SMILEScopy InChI
Affinity DataKd:  9.95E+3nMAssay Description:Binding affinity to recombinant human AMPK alpha1/beta1/gamma1 by SPR binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5BRCPubMed