Compile Data Set for Download or QSAR
Found 9 of kd for UniProtKB: P11274
LigandPNGBDBM50459091(ABL-001 | ABL001 | ABL001-NX | Asciminib | NVP-ABL...)copy SMILEScopy InChI
Affinity DataKd:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028WJ8PubMed
LigandPNGBDBM50328136(6-(1H-pyrazol-4-yl)-N-(4-(trifluoromethoxy)phenyl)...)copy SMILEScopy InChI
Affinity DataKd:  43nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50328138((4-methylpiperazin-1-yl)(4-(4-(trifluoromethoxy)ph...)copy SMILEScopy InChI
Affinity DataKd:  46nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50328137(6-(1-methyl-1H-pyrazol-4-yl)-N-(4-(trifluoromethox...)copy SMILEScopy InChI
Affinity DataKd:  57nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50325999(3-(6-(4-(trifluoromethoxy)phenylamino)pyrimidin-4-...)copy SMILEScopy InChI
Affinity DataKd:  92nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50328135(CHEMBL1257308 | N-(4-(6-(4-(trifluoromethoxy)pheny...)copy SMILEScopy InChI
Affinity DataKd:  114nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50328125(1-(pyridin-4-ylmethyl)-N-(4-(trifluoromethoxy)phen...)copy SMILEScopy InChI
Affinity DataKd:  394nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50328126(1-((2,4-dimethylthiazol-5-yl)methyl)-N-(4-(trifluo...)copy SMILEScopy InChI
Affinity DataKd:  526nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed
LigandPNGBDBM50328122(4-((4-(4-(trifluoromethoxy)phenylamino)-1H-pyrazol...)copy SMILEScopy InChI
Affinity DataKd:  598nMAssay Description:Inhibition of Bcr-Abl in mouse BA/F3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FTWPubMed