Compile Data Set for Download or QSAR
Found 123 of kd for UniProtKB: P05067
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50481603(CHEMBL607562)copy SMILEScopy InChI
Affinity DataKd:  0.210nMAssay Description:Displacement of [125I-N-Methyl-4-(4-bromoanilino)phthalimide from beta-amyloid plaques isolated from Alzheimer's disease patient brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445Q9VPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50497728(CHEMBL3314344)copy SMILEScopy InChI
Affinity DataKd:  0.560nMAssay Description:Binding affinity to amyloid beta42 (unknown origin) after 3 hrs by gamma countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1065NPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598562(CHEMBL5207165)copy SMILES
Affinity DataKd:  1.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50173647((E)-4-(4-(methylamino)styryl)phenol | 4-(4-(methyl...)copy SMILEScopy InChI
Affinity DataKd:  2.40nMAssay Description:Binding affinity to Beta amyloid aggregates in Alzheimer's disease patient brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9FW6PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598552(CHEMBL5186511)copy SMILES
Affinity DataKd:  3.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598552(CHEMBL5186511)copy SMILES
Affinity DataKd:  3.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50485997(CHEMBL2203379)copy SMILEScopy InChI
Affinity DataKd:  4.5nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19RGPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50486005(CHEMBL2203394)copy SMILEScopy InChI
Affinity DataKd:  6.40nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19RGPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50129793(2-(4''-methylaminophenyl)-6-hydroxybenzothiazole |...)copy SMILEScopy InChI
Affinity DataKd:  7.20nMAssay Description:Binding affinity to beta amyloid plaque in human Alzheimer's disease brain tissueMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2RSQPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50481119(AZD-2184 | CHEMBL570378)copy SMILEScopy InChI
Affinity DataKd:  8.40nMAssay Description:Displacement of [3H]PIB from human amyloid beta (1 to 40) fibrils after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XCMPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50485994(CHEMBL2203385)copy SMILEScopy InChI
Affinity DataKd:  9.60nMAssay Description:Displacement of [3H]DMAB from amyloid beta plaque in cortex homogenate isolated from Alzheimer disease patient after 90 mins by scintillation countin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19RGPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598567(CHEMBL5199963)copy SMILES
Affinity DataKd:  15nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598551(CHEMBL5169704)copy SMILES
Affinity DataKd:  16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598551(CHEMBL5169704)copy SMILES
Affinity DataKd:  24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598566(CHEMBL5192359)copy SMILES
Affinity DataKd:  24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50515566(CHEMBL4475538)copy SMILEScopy InChI
Affinity DataKd:  25nMAssay Description:Binding affinity to amyloid beta 1 to 42 (unknown origin) in PBS buffer at pH 7.4 assessed as binding constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB1B75PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598551(CHEMBL5169704)copy SMILES
Affinity DataKd:  27nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598556(CHEMBL5174620)copy SMILES
Affinity DataKd:  27nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50515565(CHEMBL4453231)copy SMILEScopy InChI
Affinity DataKd:  35nMAssay Description:Binding affinity to amyloid beta 1 to 42 (unknown origin) in PBS buffer at pH 7.4 assessed as binding constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB1B75PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598552(CHEMBL5186511)copy SMILES
Affinity DataKd:  38nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598536(CHEMBL5183943)copy SMILES
Affinity DataKd:  39nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484502(CHEMBL1926768)copy SMILEScopy InChI
Affinity DataKd:  42nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50515568(CHEMBL4570231)copy SMILEScopy InChI
Affinity DataKd:  46nMAssay Description:Binding affinity to amyloid beta 1 to 42 (unknown origin) in PBS buffer at pH 7.4 assessed as binding constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB1B75PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598550(CHEMBL5183307)copy SMILES
Affinity DataKd:  46nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50490495(CHEMBL2326893)copy SMILEScopy InChI
Affinity DataKd:  48nMAssay Description:Binding affinity to amyloid beta aggregate (unknown origin) by centrifugation methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0XD0PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614044(CHEMBL5283353)copy SMILES
Affinity DataKd:  48nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598553(CHEMBL5207355)copy SMILES
Affinity DataKd:  52nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598553(CHEMBL5207355)copy SMILES
Affinity DataKd:  69nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50515567(CHEMBL4524664)copy SMILEScopy InChI
Affinity DataKd:  77nMAssay Description:Binding affinity to amyloid beta 1 to 42 (unknown origin) in PBS buffer at pH 7.4 assessed as binding constant by fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB1B75PubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598553(CHEMBL5207355)copy SMILES
Affinity DataKd:  86nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484498(CHEMBL1926769)copy SMILEScopy InChI
Affinity DataKd:  91nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598550(CHEMBL5183307)copy SMILES
Affinity DataKd:  106nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598564(CHEMBL5193352)copy SMILES
Affinity DataKd:  106nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598549(CHEMBL594574)copy SMILES
Affinity DataKd:  110nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50598548(CHEMBL594555)copy SMILES
Affinity DataKd:  120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X92GCKPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484499(CHEMBL1926770)copy SMILEScopy InChI
Affinity DataKd:  167nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484500(CHEMBL1926775)copy SMILEScopy InChI
Affinity DataKd:  192nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50129784(4-(6-Methoxybenzo[d]thiazol-2-yl)-N,N-dimethylanil...)copy SMILEScopy InChI
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614053(CHEMBL5283075)copy SMILES
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614052(CHEMBL5266905)copy SMILES
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614055(CHEMBL5279844)copy SMILES
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614054(CHEMBL5281010)copy SMILES
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50614051(CHEMBL5288007)copy SMILES
Affinity DataKd:  220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484501(CHEMBL1926771)copy SMILEScopy InChI
Affinity DataKd:  222nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM195591(US9216974,Resorufin | US9333197, Resorufin)copy SMILEScopy InChI
Affinity DataKd:  225nMAssay Description:To determine the Ki values, fixed brain tissues prepared from 15-month-old Tg2576 mice (N=5) will be incubated for 30 min with 1 μM methoxy-X34 ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WD3ZCGUS Patent
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50103964(CHEMBL3593932)copy SMILEScopy InChI
Affinity DataKd:  271nMAssay Description:Binding affinity amyloid beta (1 to 42) (unknown origin) expressed in Escherichia coli after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WRCPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484504(CHEMBL1926773)copy SMILEScopy InChI
Affinity DataKd:  278nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50484503(CHEMBL1926774)copy SMILEScopy InChI
Affinity DataKd:  286nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM512913(US11091444, Compound FAH-3 | US11142505, FAH #3)copy SMILES
Affinity DataKd:  300nMAssay Description:β-sectretase inhibitor IV from Calbiochem (cat #565788).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8PVFUS Patent
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50100134(2-(4-Dimethylamino-phenyl)-3,6-dimethyl-benzothiaz...)copy SMILEScopy InChI
Affinity DataKd:  384nMAssay Description:Binding affinity to human amyloid beta (1 to 42) fibril by fluorescence intensity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QTNPubMed
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