Compile Data Set for Download or QSAR
Found 12 of kd for UniProtKB: P00523
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM50587782(CHEMBL5209202)copy SMILES
Affinity DataKd:  0.280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q5115PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 6.30nM Kd:  8nMAssay Description:Tyrosine kinase inhibition assay using wild type cSrc measured by a fluorescence-labeled approach.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8B46PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM81374(BODIPY-labeled probe, 4a)copy SMILEScopy InChI
Affinity DataKd:  11nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833QG7PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nM Kd:  11nMAssay Description:Tyrosine kinase inhibition assay using wild type cSrc measured by a fluorescence-labeled approach.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM13216(BMS-354825 | CHEMBL1421 | DASATINIB | N-(2-Chloro-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nM Kd:  11nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM81374(BODIPY-labeled probe, 4a)copy SMILEScopy InChI
Affinity DataIC50: 25.4nM Kd:  13nMpH: 7.5Assay Description:In vitro activity assay using various kinases.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833QG7PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM31829(RL46 | quinazoline-pyrazolourea hybrid compound, 3...)copy SMILEScopy InChI
Affinity DataIC50: 14nM Kd:  56nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1QD3PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM31828(quinazoline-pyrazolourea hybrid compound, 3b)copy SMILEScopy InChI
Affinity DataIC50: 21nM Kd:  73nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM31827(quinazoline-pyrazolourea hybrid compound, 3a)copy SMILEScopy InChI
Affinity DataIC50: 71nM Kd:  174nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1QD3PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM31831(quinazoline-pyrazolourea hybrid compound, 3e)copy SMILEScopy InChI
Affinity DataIC50: 235nM Kd:  239nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1QD3PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM31830(quinazoline-pyrazolourea hybrid compound, 3d)copy SMILEScopy InChI
Affinity DataIC50: 207nM Kd:  256nMpH: 7.0 T: 2°CAssay Description:IC50 determinations for cSrc kinases were measured with the HTRF KinEASE-TK assay from Cisbio according to the manufacturer instructions. A biotinyla...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1QD3PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))TBA
LigandPNGBDBM50142887(1-(tert-butyl)-3-(4-chlorophenyl)-4-aminopyrazolo[...)copy SMILEScopy InChI
Affinity DataKd:  296nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q5115PubMed