Compile Data Set for Download or QSAR
Found 9 of kd for UniProtKB: P54829
LigandPNGBDBM50583252(CHEMBL5077745)copy SMILES
Affinity DataKd:  230nMAssay Description:Inhibition of TAM-3Y-F2Pmp peptide binding to N-terminal His6-fused STEP32 (282 to 563 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0K1VPubMed
LigandPNGBDBM50583254(CHEMBL5077972)copy SMILES
Affinity DataKd:  400nMAssay Description:Inhibition of TAM-3Y-F2Pmp peptide binding to N-terminal His6-fused STEP32 (282 to 563 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0K1VPubMed
LigandPNGBDBM50583255(CHEMBL5090224)copy SMILES
Affinity DataKd:  450nMAssay Description:Inhibition of TAM-3Y-F2Pmp peptide binding to N-terminal His6-fused STEP32 (282 to 563 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0K1VPubMed
LigandPNGBDBM50583232(CHEMBL5083288)copy SMILES
Affinity DataKd:  670nMAssay Description:Inhibition of TAM-3Y-F2Pmp peptide binding to N-terminal His6-fused STEP32 (282 to 563 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0K1VPubMed
LigandPNGBDBM50441297(CHEMBL2431664 | CHEMBL2431666)copy SMILEScopy InChI
Affinity DataKd:  2.72E+4nMAssay Description:Binding affinity to 6His-tagged STEP phosphatase domain (258 to 539 residues) (unknown origin) expressed in Escherichia coli BL21 Gold (DE3) after 90...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8B27PubMed
LigandPNGBDBM50441296(CHEMBL2431665 | CHEMBL2431667)copy SMILEScopy InChI
Affinity DataKd:  3.14E+4nMAssay Description:Binding affinity to 6His-tagged STEP phosphatase domain (258 to 539 residues) (unknown origin) expressed in Escherichia coli BL21 Gold (DE3) after 90...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8B27PubMed
LigandPNGBDBM50503349(CHEMBL4476817)copy SMILEScopy InChI
Affinity DataKd:  3.80E+4nMAssay Description:Binding affinity to human 15N-labeled STEP PTP domain (281 to 563 residues) expressed in Escherichia coli OD2 by 1H,15N TROSY NMR spectral analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM50441298(CHEMBL2431708)copy SMILEScopy InChI
Affinity DataKd:  7.04E+4nMAssay Description:Binding affinity to 6His-tagged STEP phosphatase domain (258 to 539 residues) (unknown origin) expressed in Escherichia coli BL21 Gold (DE3) after 90...More data for this Ligand-Target Pair
LigandPNGBDBM50503349(CHEMBL4476817)copy SMILEScopy InChI
Affinity DataKd:  8.00E+5nMAssay Description:Binding affinity to human STEP PTP domain (281 to 563 residues) expressed in Escherichia coli BL21(DE3) by ITCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB