Compile Data Set for Download or QSAR
Found 19 of kd for UniProtKB: P29375
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245000(CHEMBL4096760)copy SMILEScopy InChI
Affinity DataKd:  60nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245002(CHEMBL4081571)copy SMILEScopy InChI
Affinity DataKd:  150nMAssay Description:Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245002(CHEMBL4081571)copy SMILEScopy InChI
Affinity DataKd:  150nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245004(CHEMBL4090351)copy SMILEScopy InChI
Affinity DataKd:  180nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245005(CHEMBL4070992)copy SMILEScopy InChI
Affinity DataKd:  210nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245037(CHEMBL4062359)copy SMILEScopy InChI
Affinity DataKd:  220nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245003(CHEMBL4066179)copy SMILEScopy InChI
Affinity DataKd:  250nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50468054(CHEMBL4284220)copy SMILEScopy InChI
Affinity DataKd:  260nMAssay Description:Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245006(CHEMBL4077310)copy SMILEScopy InChI
Affinity DataKd:  410nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50245001(CHEMBL4059617)copy SMILEScopy InChI
Affinity DataKd:  470nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM320423(2-[(2-chlorophenyl)-propoxy- methyl]-1H-pyrrolo[3,...)copy SMILES
Affinity DataKd:  530nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50282115(CHEMBL4165111)copy SMILEScopy InChI
Affinity DataKd:  800nMAssay Description:Inhibition of JARID1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G3GPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50282162(CHEMBL4173016)copy SMILEScopy InChI
Affinity DataKd:  800nMAssay Description:Inhibition of JARID1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76G3GPubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM281089(US10022354, Example 29)copy SMILEScopy InChI
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM223320(KDOAM-25)copy SMILEScopy InChI
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50468052(CHEMBL4283844)copy SMILEScopy InChI
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM50468053(CHEMBL4294426)copy SMILEScopy InChI
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM60875(3-((6-(4,5-Dihydro-1H-benzo[d]azepin-3(2H)-yl)-2-(...)copy SMILEScopy InChI
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center

Curated by ChEMBL
LigandPNGBDBM281088(US10022354, Example 28)copy SMILEScopy InChI
Affinity DataKd: >1.20E+4nMAssay Description:Binding affinity to ARID/PHD1/Zn binding domain truncated human N-terminal His-SUMO-tagged KDM5A (1 to 588 residues) expressed in Escherichia coli by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC41Z0PubMed