Compile Data Set for Download or QSAR
Found 6 of kd for UniProtKB: P55055
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50515036(CHEMBL4584267)copy SMILEScopy InChI
Affinity DataKd:  49nMAssay Description:Binding affinity to recombinant human LXRbeta-LBD expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant incubated for 30 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC42WHPubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50515025(CHEMBL4464514)copy SMILEScopy InChI
Affinity DataKd:  92nMAssay Description:Binding affinity to recombinant human LXRbeta-LBD expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant incubated for 30 mins by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC42WHPubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)copy SMILEScopy InChI
Affinity DataKd:  103nMAssay Description:Binding affinity to human LXRbeta-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50461063(CHEMBL4226803 | US10457637, Compound 8)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Activity at LXRbeta (unknown origin) expressed in human HeLa-derived HG5LN cells transfected with the GAL4 DNA-binding domain fused to the LXRbeta li...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WD437QPubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50203462(CHEMBL3931161)copy SMILEScopy InChI
Affinity DataKd: >1.00E+4nMAssay Description:Activity at GAL4 DBD-fused LXRbeta LBD (unknown origin) expressed in human HG5LN cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79DDHPubMed
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Sun Yat-sen University

Curated by ChEMBL
LigandPNGBDBM50241503(2-(3,4-Dihydroxyphenyl)-3,5,7-trihydroxy-1-Benzopy...)copy SMILEScopy InChI
Affinity DataKd:  7.32E+4nMAssay Description:Binding affinity to human LXRbeta-LBD by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3GF4PubMed