Compile Data Set for Download or QSAR
Found 107 Enz. Inhib. hit(s) with all data for entry = 50033205
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559235(CHEMBL4760126)copy SMILES
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559246(CHEMBL4752999)copy SMILES
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 2.40E+3nMAssay Description:Binding affinity to human CAMKK2 incubated for 2 hrs by nano-BRET assay based cellular target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559234(CHEMBL4781408)copy SMILES
Affinity DataIC50: 2.90E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354540(CHEMBL1836717)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human STK17A in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human CAMKK1 in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetAurora kinase B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human AURKB in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559232(CHEMBL4740090)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559236(CHEMBL4796519)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559237(CHEMBL4747753)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354559(CHEMBL1836724)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559248(CHEMBL4759004)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559238(CHEMBL4793795)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559249(CHEMBL4753500)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559250(CHEMBL4799235)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559239(CHEMBL4794226)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559245(CHEMBL4740604)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559251(CHEMBL4756902)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559252(CHEMBL4754574)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559253(CHEMBL4763345)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559254(CHEMBL4745289)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354555(CHEMBL1836637)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559255(CHEMBL4761540)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559256(CHEMBL4782453)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to C-terminal nano-luciferase tagged STK17B (unknown origin) expressed in HEK293 cells incubated for 2 hrs by nano-BRET assay based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of STK17A (unknown origin) incubated for 90 mins by Kinase seeker split luciferase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human MET in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase Nek6(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human NEK6 in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PIM2 in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human WEE1 in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CAMKK2 in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 38-like(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human STK38L in presence of ATP at Km levelMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetAurora kinase B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human AURKB incubated for 2 hrs by nano-BRET assay based cellular target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 38-like(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human STK38L incubated for 2 hrs by nano-BRET assay based cellular target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to human STK17A incubated for 2 hrs by nano-BRET assay based cellular target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataKd:  9.80E+3nMAssay Description:Binding affinity to STK17A (unknown origin) by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataKd:  440nMAssay Description:Binding affinity to human STK17A assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50354542(CHEMBL1836721)copy SMILEScopy InChI
Affinity DataKd:  270nMAssay Description:Binding affinity to STK17A (unknown origin) by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50354565(CHEMBL1836719)copy SMILEScopy InChI
Affinity DataKd:  230nMAssay Description:Binding affinity to STK17A (unknown origin) by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataKd:  910nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataKd:  5.60nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354560(CHEMBL1836641)copy SMILEScopy InChI
Affinity DataKd:  30nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354542(CHEMBL1836721)copy SMILEScopy InChI
Affinity DataKd:  11nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354565(CHEMBL1836719)copy SMILEScopy InChI
Affinity DataKd:  3.80nMAssay Description:Binding affinity to N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli by KINOMEscan scan...More data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50559221(CHEMBL4763392)copy SMILES
Affinity DataKd:  290nMAssay Description:Binding affinity to human HIPK4 by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human MET assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase Nek6(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human NEK6 assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataKd:  1.50E+3nMAssay Description:Binding affinity to human PIM2 assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
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