Compile Data Set for Download or QSAR
Found 471 of ki data for polymerid = 4981
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319615(1-(4-(4-(4-(4-Methyl-2-(methylamino)thiazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  9.70nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319623(4-(2,4-Dimethylthiazol-5-yl)-N-(3,4,5-trimethoxyph...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of CDK9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319615(1-(4-(4-(4-(4-Methyl-2-(methylamino)thiazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319627(1-(4-(4-(4-(2,4-Dimethylthiazol-5-yl)pyrimidin-2-y...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319617(CHEMBL1084630 | N-Ethyl-4-methyl-5-(2-(4-morpholin...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81438(CDK Inhibitor, 11)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM8066(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 37 | 4...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423754(CHEMBL598992)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319625(CHEMBL1083150 | N1-(4-(2,4-Dimethylthiazol-5-yl)py...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319626(4-(2,4-Dimethylthiazol-5-yl)-N-(4-(4-(methylsulfon...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319618(CHEMBL1084629 | N,4-Dimethyl-5-(2-(4-morpholinophe...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423755(CHEMBL609322)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81431(CDK Inhibitor, 4)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319615(1-(4-(4-(4-(4-Methyl-2-(methylamino)thiazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Inhibition of CDK4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81430(CDK Inhibitor, 3)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81432(CDK Inhibitor, 5)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81440(CDK Inhibitor, 13)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319624(Aminopyrimidine, 4 | CHEMBL1084454 | N1-(4-(2,4-Di...)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319620(CHEMBL1084715 | N-(4-(4-(2-(Ethylamino)-4-methylth...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423756(CHEMBL611995)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81431(CDK Inhibitor, 4)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319625(CHEMBL1083150 | N1-(4-(2,4-Dimethylthiazol-5-yl)py...)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319620(CHEMBL1084715 | N-(4-(4-(2-(Ethylamino)-4-methylth...)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Inhibition of CDK4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibition of FLT3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81435(CDK Inhibitor, 8)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81434(CDK Inhibitor, 7)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423756(CHEMBL611995)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Inhibition of CDK4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81429(CDK Inhibitor, 2)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  57nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81440(CDK Inhibitor, 13)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423757(CHEMBL609915)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81430(CDK Inhibitor, 3)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81441(CDK Inhibitor, 14)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of CDK7More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi:  73nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423758(CHEMBL598994)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81433(CDK Inhibitor, 6)copy SMILEScopy InChI
Affinity DataKi:  86nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81433(CDK Inhibitor, 6)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81433(CDK Inhibitor, 6)copy SMILEScopy InChI
Affinity DataKi:  94nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423759(CHEMBL598166)copy SMILEScopy InChI
Affinity DataKi:  98nMAssay Description:inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81439(CDK Inhibitor, 12)copy SMILEScopy InChI
Affinity DataKi:  102nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81431(CDK Inhibitor, 4)copy SMILEScopy InChI
Affinity DataKi:  107nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University of St. Andrews

Curated by ChEMBL
LigandPNGBDBM50423760(CHEMBL599804)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:inhibition of CDK9/CyclinT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81432(CDK Inhibitor, 5)copy SMILEScopy InChI
Affinity DataKi:  127nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
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