Compile Data Set for Download or QSAR
Found 28 Enz. Inhib. hit(s) with all data for entry = 10178
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518556((S)-2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-y...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518527(2-Alyl-6-((2′,3′-dihydro-1′H-spi...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518528(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518529(6-((2′-Acetyl-2′,3′-dihydro-1...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518530(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518531(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518532(2-Allyl-6-((2-ethyl-1,2,3,4-tetrahydroisoquinolin-...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518533(6-((2-Acetyl-1,2,3,4-tetrahydroisoquinolin-7-yl)am...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518534(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518535(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518536(2-Allyl-6-((4,4-dimethyl-1,2,3,4-tetrahydroisoquin...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518537(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518538(2-Allyl-6-((2-(2-hydroxyethyl)-1,2,3,4-tetrahydroi...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518539(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518540(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518541(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518542(7-((2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-y...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518546(7-((2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-y...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518547(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518549(2-allyl-6-((2-(dimethylamino)-2,3-dihydro-1H-inden...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518550(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518526(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518555((R)-2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-y...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518552(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518554(2-Allyl-6-((4,4-difluoro-1,2,3,4-tetrahydroisoquin...)copy SMILES
Affinity DataIC50: 10nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518553(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 55nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent
TargetWee1-like protein kinase(Homo sapiens (Human))TBA
LigandPNGBDBM518551(2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-6...)copy SMILES
Affinity DataIC50: 55nMAssay Description:Wee 1 kinase was determined by using Flurorescence Resonance Energy Transfer (FRET) assay. In 384-well plates, Wee1 kinase (2 nM final concentration)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R214JBUS Patent