Compile Data Set for Download or QSAR
Found 237 Enz. Inhib. hit(s) with all data for entry = 2628
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311218((S)-1-(2-cyclopropyl-4-(quinolin-4-yl)phenoxy)-2,4...)copy SMILEScopy InChI
Affinity DataIC50: 0.0700nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311290((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 0.190nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311339((S)-methyl (6-((2-amino-2,4-dimethylpentyl)oxy)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311347((S)-1-((3-(difluoromethyl)-5-(quinolin-4-yl)pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311289((S)-2,4-dimethyl-1-((6-(quinolin-4-yl)-4-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 0.240nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311338((S)-1-((3-(difluoromethyl)-5-(7-fluoroquinolin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311155((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-cyanop...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311265((S)-1-((4-(difluoromethyl)-6-(quinolin-4-yl)pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311340((S)-1-((5-(7-chloroquinolin-4-yl)-3-(difluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311229((S)-1-(4-(1,6-naphthyridin-4-yl)-2-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311189((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311292((S)-1-((4-(difluoromethyl)-5′-fluoro-2′...)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311176((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311170((S)-N-(4-(4-((2-amino-2,4-dimethylpentyl)oxy)-3-(t...)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311378((S)-1-((4-chloro-6-(6-fluoroquinolin-4-yl)pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311206((S)-1-(2-(difluoromethyl)-4-(2-methylpyridin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311363((S)-methyl (6-((2-amino-2,4-dimethylpentyl)oxy)-5-...)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311382((S)-1-((4-chloro-6-(6-chloroquinolin-4-yl)pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311370((S)-1-((6-(7-fluoroquinolin-4-yl)-4-methylpyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.410nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311159((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311287((S)-1-((2′-chloro-4-(difluoromethyl)-5′...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311232((S)-1-(4-(7-chloroquinolin-4-yl)-2-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.460nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311158((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-(trifl...)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311374((S)-1-((6-(7-chloroquinolin-4-yl)-4-methylpyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM373597((S)-1-((3-chloro-5-(quinolin-4-yl)pyridin-2-yl)oxy...)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311332((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-fluoro...)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311157((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-(trifl...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311264((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311217((S)-1-(4-(6-fluoroquinolin-4-yl)-2-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311193((S)-1-(2-(difluoromethyl)-4-(2-(difluoromethyl)pyr...)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311266((S)-1-((4-(difluoromethyl)-2′-methyl-[2,4...)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311160((S)-N-(4-(4-((2-amino-4-methylpentyl)oxy)-3-chloro...)copy SMILEScopy InChI
Affinity DataIC50: 0.530nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311216((S)-1-(4-(5,7-difluoroquinolin-4-yl)-2-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 0.530nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311215((S)-1-(4-(7-fluoroquinolin-4-yl)-2-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.550nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311360((S)-1-(4-(6-chloroquinolin-4-yl)-2-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 0.560nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311291((S)-1-((2′-chloro-4-(difluoromethyl)-[2,4...)copy SMILEScopy InChI
Affinity DataIC50: 0.560nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311362((S)-2,4-dimethyl-1-((5-(quinolin-4-yl)-3-(trifluor...)copy SMILEScopy InChI
Affinity DataIC50: 0.590nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM373626((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.620nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311180((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.630nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311344((S)-1-((3-(difluoromethyl)-5-(5,7-difluoroquinolin...)copy SMILEScopy InChI
Affinity DataIC50: 0.640nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311199((S)-2,4-dimethyl-1-(4-(pyridin-4-yl)-2-(trifluorom...)copy SMILEScopy InChI
Affinity DataIC50: 0.640nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311210((S)-methyl (5-((2-amino-2,4-dimethylpentyl)oxy)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311178((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM373608((S)-4-(4-((2-amino-2,4-dimethylpentyl)oxy)-3-(trif...)copy SMILEScopy InChI
Affinity DataIC50: 0.660nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM373556(US9902722, Example 29 | methyl (4-(4-((2-amino-2,4...)copy SMILEScopy InChI
Affinity DataIC50: 0.670nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311247((S)-2-((2-amino-2,4-dimethylpentyl)oxy)-5-(3-fluor...)copy SMILEScopy InChI
Affinity DataIC50: 0.680nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311295((S)-1-(2-(difluoromethyl)-4-(2-methylpyrimidin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.680nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311182((S)-methyl (4-(4-((2-amino-2,4-dimethylpentyl)oxy)...)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311348((S)-1-((3-(difluoromethyl)-5-(7-methylquinolin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
TargetAP2-associated protein kinase 1(Homo sapiens (Human))
University of Mississippi

LigandPNGBDBM311249((S)-2-((2-amino-2,4-dimethylpentyl)oxy)-5-(5-fluor...)copy SMILEScopy InChI
Affinity DataIC50: 0.720nMAssay Description:The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2930WGGUS Patent
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