Compile Data Set for Download or QSAR
Found 477 Enz. Inhib. hit(s) with all data for entry = 2817
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381327(4-chloro-1-(4-methoxy-butyl)-3- methyl-1H-pyrazolo...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381334(4-Chloro-3-methyl-1-(tetrahydro- pyran-4-yl)-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381335(4-Chloro-3-methyl-1-(tetrahydro- pyran-4-yl)-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381336(4-Chloro-3-methyl-1-(tetrahydro- pyran-4-yl)-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381339(4-chloro-1-(1-ethyl-piperidin-4-yl)- 3-methyl-1H-p...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381340(4-chloro-1-(1-ethyl-piperidin-4-yl)- 3-methyl-1H-p...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381344(4-chloro-3-methyl-1-(1- methylpiperidin-4-yl)-N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381345(4-chloro-N-(4-chlorophenyl)-3- methyl-1-(1-methylp...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381346(4-chloro-N-(4-isopropylphenyl)-3- methyl-1-(1-meth...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381353(1-(1-benzylpiperidin-4-yl)-4- chloro-3-methyl-N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381360(1-(1-acetylpiperidin-4-yl)-4-chloro- 3-methyl-N-(4...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381365(4-chloro-N-(4-isopropylphenyl)-3- methyl-1-(tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381366(4-chloro-3-methyl-1-(tetrahydro- 2H-thiopyran-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381367(4-chloro-1-(1,1-dioxidotetrahydro- 2H-thiopyran-4-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381368(4-chloro-N-(4-chlorophenyl)-1- (1,1-dioxidotetrahy...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381369(4-chloro-1-(1,1-dioxidotetrahydro- 2H-thiopyran-4-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381372(4-Chloro-1-(1-isopropyl-piperidin- 4-yl)-1H-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381373(4-Chloro-1-(1-ethyl-piperidin-4- yl)-1H-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381374(4-chloro-1-(1-ethyl-piperidin-4-yl)- 1H-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381376(4-chloro-1-(1-methyl-piperidin-4- yl)-1H-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381377(4-chloro-1-(1-methyl-piperidin-4- yl)-1H-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381378(4-Chloro-1-(tetrahydro-pyran-4- yl)-1H-pyrazolo[3,...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381379(4-Chloro-1-(tetrahydro-pyran-4- yl)-1H-pyrazolo[3,...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381380(4-chloro-N-(4-isopropylphenyl)-1- (tetrahydro-2H-p...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381387(4-Chloro-3-fluoro-1-(tetrahydro- pyran-4-yl)-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381388(4-Chloro-3-fluoro-1-(tetrahydro- pyran-4-yl)-1H-py...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381390(4-chloro-1-(tetrahydro-2H- thiopyran-4-yl)-N-(4- (...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381391(4-chloro-N-(4-isopropylphenyl)-1- (tetrahydro-2H-t...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381396(4-chloro-1-(1,1-dioxidotetrahydro- 2H-thiopyran-4-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381397(4-chloro-1-(1,1-dioxidotetrahydro- 2H-thiopyran-4-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381398(4-chloro-N-(4-chlorophenyl)-3- methyl-1-(pyridin-4...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381399(4-chloro-3-methyl-1-(pyridin-4- ylmethyl)-N-(4- (t...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381400(4-chloro-N-(4-isopropylphenyl)-3- methyl-1-(pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381413(4-Chloro-3-methyl-1-(6-methyl- pyridin-3-methyl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381414(4-Chloro-1-(5-methoxy-pyridin-2- ylmethyl)-3-methy...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381415(4-Chloro-1-(5-methoxy-pyridin-2- ylmethyl)-3-methy...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381435(4-Chloro-3-methyl-1-(5-methyl- thiazol-2-ylmethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381436(4-Chloro-3-methyl-1-(5-methyl- thiazol-2-ylmethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381439(4-chloro-N-(4-chlorophenyl)-1-((1- ethyl-1H-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381440(4-chloro-1-((1-ethyl-1H-imidazol- 2-yl)methyl)-3-m...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381442(4-chloro-1-((1-isopropyl-1H- imidazol-2-yl)methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381447(4-chloro-1-(pyridin-4-ylmethyl)-N-(4-(trifluoromet...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381448(4-chloro-N-(4-isopropylphenyl)-1-(pyridin-4-ylmeth...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381450(4-chloro-1-(pyridin-3-ylmethyl)-N-(4-(trifluoromet...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381451(4-chloro-N-(4-isopropylphenyl)-1-(pyridin-3-ylmeth...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381453(4-chloro-1-(pyridin-2-ylmethyl)-N-(4-(trifluoromet...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381454(4-chloro-N-(4-isopropylphenyl)-1-(pyridin-2-ylmeth...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381464(4-chloro-N-(4-isopropylphenyl)-1- ((1-methyl-1H-im...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381467(4-chloro-1-((1-methyl-1H- imidazol-2-yl)methyl)-N-...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
TargetGlucocorticoid receptor(Homo sapiens (Human))
GlaxoSmithKline

LigandPNGBDBM381468(4-chloro-N-(4-isopropylphenyl)-1- ((1-methyl-1H-im...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The assay was performed using H4 neuroglioma cells and using indirect immunofluorescence detection of the endogenous GR receptor. Fixative: 4% PFA. P...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29P33Z7US Patent
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