Compile Data Set for Download or QSAR
Found 68 Enz. Inhib. hit(s) with all data for entry = 50000003
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239059(CHEMBL4059503)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239059(CHEMBL4059503)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239059(CHEMBL4059503)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239056(CHEMBL4062264)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239062(CHEMBL4088364)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220250(US9290476, 95)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220220(US9290476, 63A | US9290476, 63B | US9290476, 63C)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239073(CHEMBL4097986)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239063(CHEMBL4094197)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220219(US9290476, 62A | US9290476, 62B | US9290476, 62C)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220192(US9290476, 35A | US9290476, 35B | US9290476, 35C)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220250(US9290476, 95)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220190(US9290476, 33A | US9290476, 33B | US9290476, 33C)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220190(US9290476, 33A | US9290476, 33B | US9290476, 33C)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220192(US9290476, 35A | US9290476, 35B | US9290476, 35C)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Compound was evaluated for binding affinity by the inhibition of Glutamine synthetase (Ovine brain) activity using biosynthetic assay [competitive in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239064(CHEMBL4073568)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239066(CHEMBL4063937)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239058(CHEMBL4100439)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239071(CHEMBL4101932)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220219(US9290476, 62A | US9290476, 62B | US9290476, 62C)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220220(US9290476, 63A | US9290476, 63B | US9290476, 63C)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239060(CHEMBL4070889)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239067(CHEMBL4072529)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239065(CHEMBL4083942)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239053(CHEMBL4071285)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239051(CHEMBL4097051)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239054(CHEMBL4098583)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239057(CHEMBL4090273)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239072(CHEMBL4091706)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239068(CHEMBL4099447)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239055(CHEMBL4101047)copy SMILEScopy InChI
Affinity DataIC50: 2.74E+3nMAssay Description:Inverse agonist activity at RORgammat in human Th17 cells assessed as inhibition of IL17A productionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239052(CHEMBL4098325)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Evaluated in vitro for inhibitory potency against renin.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239054(CHEMBL4098583)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239070(CHEMBL4082428)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239055(CHEMBL4101047)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239061(CHEMBL4083071)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inverse agonist activity at GAL4 DBD-fused human RORgammat expressed in HEK293T cells assessed as inhibition of transcriptional activity after 24 hrs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239052(CHEMBL4098325)copy SMILEScopy InChI
Affinity DataKd:  1.00E+4nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239053(CHEMBL4071285)copy SMILEScopy InChI
Affinity DataKd:  160nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220190(US9290476, 33A | US9290476, 33B | US9290476, 33C)copy SMILEScopy InChI
Affinity DataKd:  9.20nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220250(US9290476, 95)copy SMILEScopy InChI
Affinity DataKd:  7.70nMAssay Description:In vitro for binding affinity against sigma receptor using [3H](+)-3-PPP as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220220(US9290476, 63A | US9290476, 63B | US9290476, 63C)copy SMILEScopy InChI
Affinity DataKd:  6.20nMAssay Description:In vitro for binding affinity against sigma receptor using [3H](+)-3-PPP as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220192(US9290476, 35A | US9290476, 35B | US9290476, 35C)copy SMILEScopy InChI
Affinity DataKd:  5nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM220219(US9290476, 62A | US9290476, 62B | US9290476, 62C)copy SMILEScopy InChI
Affinity DataKd:  1.5nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239061(CHEMBL4083071)copy SMILEScopy InChI
Affinity DataKd:  20nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239069(CHEMBL4079036)copy SMILEScopy InChI
Affinity DataKd:  37nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239051(CHEMBL4097051)copy SMILEScopy InChI
Affinity DataKd:  32nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239060(CHEMBL4070889)copy SMILEScopy InChI
Affinity DataKd:  15nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239070(CHEMBL4082428)copy SMILEScopy InChI
Affinity DataKd:  9.50E+3nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239057(CHEMBL4090273)copy SMILEScopy InChI
Affinity DataKd:  1.50E+4nMAssay Description:In vitro for binding affinity against sigma receptor using [3H](+)-3-PPP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50239056(CHEMBL4062264)copy SMILEScopy InChI
Affinity DataKd:  2nMAssay Description:Displacement of 1,8-ANS from recombinant human RORgammat LBD expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of co-activator SR...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7JCJPubMed
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