Compile Data Set for Download or QSAR
Found 69 Enz. Inhib. hit(s) with all data for entry = 50000100
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233444(CHEMBL4061083)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240582(CHEMBL4081380)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240581(CHEMBL4099401)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240580(CHEMBL4070782)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240585(CHEMBL4070631)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240580(CHEMBL4070782)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240584(CHEMBL4073517)copy SMILEScopy InChI
Affinity DataIC50: 148nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240577(CHEMBL4096950)copy SMILEScopy InChI
Affinity DataIC50: 188nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate pretreated for 10 mins followed by substrate addition measured after 10 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 970nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240583(CHEMBL4085712)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate pretreated for 10 mins followed by substrate addition measured after...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240582(CHEMBL4081380)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240583(CHEMBL4085712)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240574(CHEMBL4064147)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233444(CHEMBL4061083)copy SMILEScopy InChI
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240585(CHEMBL4070631)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate pretreated for 10 mins followed by substrate addition measured after 10 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240574(CHEMBL4064147)copy SMILEScopy InChI
Affinity DataIC50: 7.40E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240581(CHEMBL4099401)copy SMILEScopy InChI
Affinity DataIC50: 9.50E+3nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatographic m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240578(CHEMBL4069755)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240578(CHEMBL4069755)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TEC using poly[Glu:Tyr] (4:1) as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatograph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human JAK3 using GEEEEYFELVKKKK as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatographic m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human FMS using poly[Glu:Tyr] (4:1) as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatograph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human VEGFR2 using poly[Glu:Tyr] (4:1) as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatogr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human BTK using KVEKIGEGTYGVVYK as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatographic m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ITK using myelin basic protein as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatograp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50233461(CHEMBL4068896)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EGFR using poly[Glu:Tyr] (4:1) as substrate measured after 120 mins in presence of [gamma33P]ATP by P81 ion exchange chromatograp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240577(CHEMBL4096950)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged FGFR1 cytoplasmic domain (308 to 731 residues) expressed in baculovirus expression system using tyr 04 as ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240573(CHEMBL4077859)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50240575(CHEMBL4089245)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M90BT6PubMed
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