Compile Data Set for Download or QSAR
Found 70 Enz. Inhib. hit(s) with all data for entry = 50000235
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242934(CHEMBL4066743)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of platelet aggregation (PRP)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242894(CHEMBL4074323)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM301063(4-{3-[((3R)-3- aminopiperidyl)carbonyl]-5-(2- pyri...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of full length human LSD1 expressed in Escherichia coli using H3K4me1-biotin labeled peptide as substrate after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242895(CHEMBL4076163)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of platelet aggregation (PRP)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242950(CHEMBL4074334)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242905(CHEMBL4103503)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242892(CHEMBL4088045)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242886(CHEMBL4104407)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM301063(4-{3-[((3R)-3- aminopiperidyl)carbonyl]-5-(2- pyri...)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242952(CHEMBL4088035)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242953(CHEMBL4066749)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242907(CHEMBL4077730)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242905(CHEMBL4103503)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242934(CHEMBL4066743)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242883(CHEMBL4062785)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242891(CHEMBL4095768)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242890(CHEMBL4077739)copy SMILEScopy InChI
Affinity DataIC50: 670nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242948(CHEMBL4082935)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242889(CHEMBL4069461)copy SMILEScopy InChI
Affinity DataIC50: 720nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242956(CHEMBL4085581)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Inhibition of Fibrinogen receptor bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242951(CHEMBL4096682)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242887(CHEMBL4080173)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242896(CHEMBL4093330)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242885(CHEMBL4101077)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242945(CHEMBL4073624)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242942(CHEMBL4092725)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242895(CHEMBL4076163)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM301063(4-{3-[((3R)-3- aminopiperidyl)carbonyl]-5-(2- pyri...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of LSD1 in human THP1 cells assessed as upregulation of CD86 levels by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242884(CHEMBL4090735)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242906(CHEMBL4095757)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242946(CHEMBL4062278)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50241539(CHEMBL4084845)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242957(CHEMBL4100451)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human ERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242943(CHEMBL4065043)copy SMILEScopy InChI
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242947(CHEMBL4083993)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242958(CHEMBL4070901)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli using Histone H3(1 to 21)K4(Me1) biotin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242952(CHEMBL4088035)copy SMILEScopy InChI
Affinity DataKd:  22nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242957(CHEMBL4100451)copy SMILEScopy InChI
Affinity DataKd:  450nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242948(CHEMBL4082935)copy SMILEScopy InChI
Affinity DataKd:  240nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242951(CHEMBL4096682)copy SMILEScopy InChI
Affinity DataKd:  240nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242907(CHEMBL4077730)copy SMILEScopy InChI
Affinity DataKd:  66nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242905(CHEMBL4103503)copy SMILEScopy InChI
Affinity DataKd:  34nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242891(CHEMBL4095768)copy SMILEScopy InChI
Affinity DataKd:  87nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242934(CHEMBL4066743)copy SMILEScopy InChI
Affinity DataKd:  6nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242954(CHEMBL4101067)copy SMILEScopy InChI
Affinity DataKd:  21nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242895(CHEMBL4076163)copy SMILEScopy InChI
Affinity DataKd:  7nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Manchester

Curated by ChEMBL
LigandPNGBDBM50242892(CHEMBL4088045)copy SMILEScopy InChI
Affinity DataKd:  32nMAssay Description:Reversible inhibition of human recombinant N-terminal truncated LSD1 (151 to 852 residues) expressed in Escherichia coli by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047W8PubMed
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