Compile Data Set for Download or QSAR
Found 48 Enz. Inhib. hit(s) with all data for entry = 50000689
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258507(CHEMBL4078345)copy SMILEScopy InChI
Affinity DataKi:  0.0380nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258514(CHEMBL4062015)copy SMILEScopy InChI
Affinity DataKi:  0.0740nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258507(CHEMBL4078345)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258506(CHEMBL4072275)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258515(CHEMBL4083754)copy SMILEScopy InChI
Affinity DataKi:  0.610nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258544(CHEMBL4096388)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258542(CHEMBL4082758)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258514(CHEMBL4062015)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258544(CHEMBL4096388)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258500(CHEMBL4093034)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258523(CHEMBL2402204)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258524(CHEMBL4081250)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258498(CHEMBL4101714)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258515(CHEMBL4083754)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258543(CHEMBL4070637)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258499(CHEMBL4100751)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258500(CHEMBL4093034)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258542(CHEMBL4082758)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258498(CHEMBL4101714)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258499(CHEMBL4100751)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258524(CHEMBL4081250)copy SMILEScopy InChI
Affinity DataKi:  45nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258541(CHEMBL4060936)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258537(CHEMBL4099269)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258506(CHEMBL4072275)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258541(CHEMBL4060936)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258543(CHEMBL4070637)copy SMILEScopy InChI
Affinity DataKi:  250nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258523(CHEMBL2402204)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetProcathepsin L(Homo sapiens (Human))
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258537(CHEMBL4099269)copy SMILEScopy InChI
Affinity DataKi:  330nMAssay Description:Inhibition of human cathepsin L using Cbz-Phe-Arg-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258492(CHEMBL4074432)copy SMILEScopy InChI
Affinity DataKi:  1.74E+3nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258544(CHEMBL4096388)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258506(CHEMBL4072275)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50157741(CHEMBL374508 | E-64 | E64)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258514(CHEMBL4062015)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258515(CHEMBL4083754)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258543(CHEMBL4070637)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258507(CHEMBL4078345)copy SMILEScopy InChI
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258523(CHEMBL2402204)copy SMILEScopy InChI
Affinity DataIC50: 7.33E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258498(CHEMBL4101714)copy SMILEScopy InChI
Affinity DataIC50: 9.53E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258499(CHEMBL4100751)copy SMILEScopy InChI
Affinity DataIC50: 9.63E+3nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258500(CHEMBL4093034)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258541(CHEMBL4060936)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258542(CHEMBL4082758)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258524(CHEMBL4081250)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258545(CHEMBL4090306)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258492(CHEMBL4074432)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed
TargetFalcipain 2(Plasmodium falciparum)
Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina , Viale Annunziata, 98168 Messina, Italy.

Curated by ChEMBL
LigandPNGBDBM50258537(CHEMBL4099269)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum falcipain-2 expressed in Escherichia coli M15(pREP4) using Cbz-Phe-Arg-AMC as substrate by fluorescen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2K73PubMed