Compile Data Set for Download or QSAR
Found 16 Enz. Inhib. hit(s) with all data for entry = 50000948
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50048908(CHEMBL415788)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265841(CHEMBL4100456)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265836(CHEMBL4084378)copy SMILEScopy InChI
Affinity DataKi:  262nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265835(CHEMBL4076517)copy SMILEScopy InChI
Affinity DataKi:  456nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265835(CHEMBL4076517)copy SMILEScopy InChI
Affinity DataKi:  474nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265842(CHEMBL4103884)copy SMILEScopy InChI
Affinity DataKi:  620nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265841(CHEMBL4100456)copy SMILEScopy InChI
Affinity DataKi:  663nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265833(CHEMBL4082440)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265834(CHEMBL4074624)copy SMILEScopy InChI
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptor expressed in human 1321N1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265836(CHEMBL4084378)copy SMILEScopy InChI
Affinity DataKi:  5.70E+3nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265834(CHEMBL4074624)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265833(CHEMBL4082440)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50265842(CHEMBL4103884)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptor expressed in CHOK1 cell membranes after 30 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50342242((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)...)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed
TargetNeurotensin receptor type 2(Homo sapiens (Human))
Universit£ Montpellier

Curated by ChEMBL
LigandPNGBDBM50342242((S)-2-((2S,3S)-2-((S)-2-((S)-1-((S)-6-amino-2-((S)...)copy SMILEScopy InChI
Affinity DataIC50: 0.950nMAssay Description:Displacement of 125I-[Tyr3]-NT from human NTS2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377C6VPubMed