TargetHistone deacetylase 3(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of HDAC3 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of HDAC6 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibition of HDAC8 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q22R3V5JPubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q22R3V5JPubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetHistone deacetylase 1(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HDAC1 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, MI 48202, United States.
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of HDAC3 (unknown origin) by ELISA-based assayMore data for this Ligand-Target Pair
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