Compile Data Set for Download or QSAR
Found 96 Enz. Inhib. hit(s) with all data for entry = 50001121
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269689(CHEMBL4075584)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269688(CHEMBL4077439)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269694(CHEMBL4088221)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269697(CHEMBL4062038)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269693(CHEMBL4062597)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269696(CHEMBL4081975)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269698(CHEMBL4093696)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269695(CHEMBL4076384)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269699(CHEMBL4076381)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269685(CHEMBL4077529)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269701(CHEMBL4078864)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269700(CHEMBL4068293)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269686(CHEMBL4077036)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269704(CHEMBL4061800)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269702(CHEMBL4061901)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269703(CHEMBL4089866)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269706(CHEMBL4088418)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269689(CHEMBL4075584)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269698(CHEMBL4093696)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269686(CHEMBL4077036)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269689(CHEMBL4075584)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269688(CHEMBL4077439)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269688(CHEMBL4077439)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269696(CHEMBL4081975)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269697(CHEMBL4062038)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269699(CHEMBL4076381)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269694(CHEMBL4088221)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269700(CHEMBL4068293)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269693(CHEMBL4062597)copy SMILEScopy InChI
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269694(CHEMBL4088221)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269701(CHEMBL4078864)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269704(CHEMBL4061800)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269685(CHEMBL4077529)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269686(CHEMBL4077036)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269695(CHEMBL4076384)copy SMILEScopy InChI
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269697(CHEMBL4062038)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269696(CHEMBL4081975)copy SMILEScopy InChI
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269698(CHEMBL4093696)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
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