Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with all data for entry = 50001210
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50143558(CHEMBL41355 | EZOGABINE | N-(2-amino-4-(4-fluorobe...)copy SMILEScopy InChI
Affinity DataEC50:  350nMAssay Description:Activation of KCNQ2 (unknown origin) expressed in CHO cells at 10 uM after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50272431(CHEMBL4126028)copy SMILEScopy InChI
Affinity DataEC50:  1.58E+3nMAssay Description:Activation of KCNQ2 (unknown origin) expressed in CHO cells at 10 uM after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CFMPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50272438(CHEMBL4128096)copy SMILEScopy InChI
Affinity DataEC50:  130nMAssay Description:Activation of KCNQ2 (unknown origin) expressed in CHO cells at 10 uM after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CFMPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50272437(CHEMBL4125892)copy SMILEScopy InChI
Affinity DataEC50:  220nMAssay Description:Activation of KCNQ2 (unknown origin) expressed in CHO cells at 10 uM after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CFMPubMed
TargetPotassium voltage-gated channel subfamily KQT member 2(Homo sapiens (Human))
Nanjing University of Technology

Curated by ChEMBL
LigandPNGBDBM50272436(CHEMBL4126113)copy SMILEScopy InChI
Affinity DataEC50:  330nMAssay Description:Activation of KCNQ2 (unknown origin) expressed in CHO cells at 10 uM after 10 mins by atomic absorption spectrophotometry-based Rb+ flow assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CFMPubMed