Found 20 Enz. Inhib. hit(s) with all data for entry = 50001367 
Affinity DataIC50: 0.300nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Binding affinity to CXCR4 in human MDA-MB-231 cells preincubated for 15 mins followed by biotinylated TN41003 addition measured after 30 mins by rhod...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-SDF-1alpha from CXCR4 in human MDA-MB-231 cells after 60 mins by gamma-counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Antagonist activity at CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Antagonist activity at CXCR4 in human MOLT-4 cells assessed as decrease in SDF-1alpha induced cytosolic Ca2+ levels preincubated for 30 mins followed...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Antagonist activity at CXCR4 in human U87-MG cells assessed as inhibition of CXCL12-induced cell proliferation after 1 hr by MTT assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.50E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.10E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+4nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced receptor activationMore data for this Ligand-Target Pair
